N-Benzylnaltrindole hydrochloride
Tocris Bioscience, part of Bio-Techne | Catalog # 0754
Selective non-peptide δ2 antagonist
Discontinued Product
0754 has been discontinued.
View all delta Opioid Receptor Antagonists products.
Key Product Details
Description
Selective non-peptide δ2 antagonist
Product Description
N-Benzylnaltrindole hydrochloride is a potent δ2-selective opioid receptor antagonist with a long duration of action in vivo.Product Specifications
Molecular Weight
541.09
Formula
C33H32N2O3.HCl
Storage
Store at RT
Chemical Name
1'-Benzyl-17-(cyclopropylmethyl)-6,7-didehydro-4,5a-epoxy-3,14-dihydroxyindolomorphinan hydrochloride
CAS Number
1206487-81-1
PubChem ID
90479740
InChI Key
KDEBSUYWJUBPCB-ZHYTUUPESA-N
SMILES
O[C@@]24[C@]3([C@@H]8C(N6CC7=CC=CC=C7)=C(C5=C6C=CC=C5)C4)C1=C(O8)C(O)=CC=C1CC2N(CC9CC9)CC3.Cl
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Solubility
| Solvent | Max Conc. mg/mL | Max Conc. mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 54.11 | 100 |
Preparing Stock Solutions
for N-Benzylnaltrindole hydrochloride
The following data is based on the product molecular weight 541.09
Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.85 mL | 9.24 mL | 18.48 mL |
| 5 mM | 0.37 mL | 1.85 mL | 3.70 mL |
| 10 mM | 0.18 mL | 0.92 mL | 1.85 mL |
| 50 mM | 0.04 mL | 0.18 mL | 0.37 mL |
Calculators
Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Background References
References are publications that support the biological activity of the product.
- Korlipara N-Benzylnaltrindoles as long acting δ-opioid receptor antagonists. J.Med.Chem. 1994 PMID: 8021928
Product Specific Notices for N-Benzylnaltrindole hydrochloride
For research use only
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