18 results for "Adenosine A1R Small Molecules and Peptides" in Products
Adenosine A1R Small Molecules and Peptides
Adenosine A1 Receptor (ADORA1, Adenosine A1R) is an adenosine receptor that belongs to the G protein-coupled receptor 1 family. There are 3 types of adenosine receptors, each with a specific pattern of ligand binding and tissue distribution, and together they regulate a diverse set of physiologic functions. The Adenosine A1R inhibits adenylyl cyclase, and plays a role in the fertilization process. Animal studies also suggest a role for A1 receptors in kidney function and ethanol intoxication.
Selective A1 antagonist
High affinity adenosine agonist
Endogenous adenosine receptor agonist
A1 and A2B antagonist. CNS stimulant
PDE inhibitor (non-selective)
Positive allosteric modulator of A1 receptors
Potent and selective A1 agonist
Potent and selective A1 agonist
Adenosine receptor agonist
Potent adenosine receptor antagonist
Potent and selective A1 agonist
Highly selective A1 agonist
Selective A1 antagonist
Adenosine receptor antagonist
Highly selective and potent A1 receptor agonist
Adenosine receptor antagonist
High affinity adenosine A1 receptor antagonist
Positive allosteric modulator (PAM) of A1 receptors; also allosteric partial agonist in absence of orthosteric agonist
