Estropipate

Name: Estropipate
Brand: Tocris Bioscience
SKU: 3588

Tocris Bioscience, part of Bio-Techne | Catalog # 3588

COA / SDS

Estrogen receptor agonist and OATP1B1 inhibitor

Discontinued Product

3588 has been discontinued. View all Estrogen and Related Receptor Agonists products.

Key Product Details

Description:	Estrogen receptor agonist and OATP1B1 inhibitor
Chemical Name:	Piperazine estrone sulfate
Purity:	≥97% (HPLC)
Molecular Weight:	436.56

View Full Technical Details for Estropipate

Technical Data
Citations

Biological Activity for Estropipate

Estrogen receptor agonist. Also inhibits organic anion transporting polypeptide 1B1 (OATP1B1) (IC₅₀= 70 nM).

Technical Data for Estropipate

M. Wt	436.56
Formula	C₁₈H₂₂O₅S.C₄H₁₀N₂
Storage	Store at RT
Purity	≥97% (HPLC)
CAS Number	7280-37-7
PubChem ID	5284555
InChi Key	HZEQBCVBILBTEP-ZFINNJDLSA-N
Smiles	O=C4CC[C@@]3([H])[C@]2([H])CCC1=CC(OS(=O)(O)=O)=CC=C1[C@]([H])2CC[C@@]34C.C5NCCNC5

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Molarity Calculator

Calculate the mass, volume, or concentration required for a solution.

Mass

Concentration

Volume

M. Wt*

g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and CoA (available online).

Dilution Calculator

Calculate the dilution required to prepare a stock solution.

Concentration 1 (C1)

Volume 1 (V1)

Concentration 2 (C2)

Volume 2 (V2)

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

Volume (to add to vial)

Mass (in vial)

Desired Reconstitution Concentration

References for Estropipate

References are publications that support the biological activity of the product.

Obaidat A cell-based high-throughput assay to identify inhibitors of organic anion transporting polypeptides 1B1 and 1B3. FASEB J.
Williams Estrogen regulation of the cytochrome P450 3A subfamily in humans. J.Pharmacol.Exp.Ther. 2004 PMID: 15282264

Product Documents for Estropipate

COA

Certificate of Analysis

To download a Certificate of Analysis, please select a batch below.

SDS

⚠ WARNING: This product can expose you to chemicals including Estropipate, which is known to the State of California to cause reproductive toxicity with developmental effects. For more information, go to www.P65Warnings.ca.gov