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40 results for "Other Kinase Inhibitors Small Molecules and Peptides" in Products

Other Kinase Inhibitors: Small Molecules and Peptides

Potent and selective Lck and Src inhibitor; also inhibits SIK

Alternate Names: KIN112
Chemical Name: 2,6-Dimethylphenyl-N-(2,4-dimethoxyphenyl)-N-[2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]carbamate
Purity: ≥98% (HPLC)
Potent and selective Lck and Src inhibitor; also inhibits SIK

CaM kinase III (eEF-2 kinase) inhibitor

Chemical Name: 1-Hexadecyl-2-methyl-3-(phenylmethyl)-1H-imidazolium iodide
CaM kinase III (eEF-2 kinase) inhibitor

Potent and selective TAK1/MAP3K7 kinase inhibitor

Chemical Name: N1-(1-Propyl-1H-benzimidazol-2-yl)-1,3-benzenedicarboxamide
Purity: ≥98% (HPLC)
Potent and selective TAK1/MAP3K7 kinase inhibitor

Potent and selective TAK1 MAPKKK inhibitor

Chemical Name: (3S,5Z,8S,9S,11E)-3,4,9,10-tetrahydro-8,9,16-trihydroxy-14-methoxy-3-methyl-1H-2-benzoxacyclotetradecin-1,7(8H)-dione
Purity: ≥98% (HPLC)
Potent and selective TAK1 MAPKKK inhibitor

Potent MSK1 inhibitor; also inhibits other AGC group kinases

Chemical Name: 2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-N-4-piperidinyl-1H-imidazo[4,5-c]pyridine-7-methanamine dihydrochloride
Purity: ≥98% (HPLC)
Potent MSK1 inhibitor; also inhibits other AGC group kinases

Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable

Chemical Name: 5,11-Dihydro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-11-methyl-5-(2,2,2-trifluoroethyl)-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one
Purity: ≥98% (HPLC)
Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable

Serum- and glucocorticoid-regulated kinase (SGK) inhibitor

Chemical Name: 2-Cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl-benzoic acid
Purity: ≥97% (HPLC)
Serum- and glucocorticoid-regulated kinase (SGK) inhibitor

Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor

Chemical Name: 4a,7a-Dihydro-2-(1-hydroxyundecyl)-1-[(4-nitrophenyl)amino]-6-phenyl-1H-pyrrolo[3,4-b]pyridine-5,7(2H,6H)-dione
Purity: ≥98% (HPLC)
Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor

Potent and selective PI 4-kinase IIIβ inhibitor

Chemical Name: N-[2-[[6-Chloro-3-[3-[(dimethylamino)sulfonyl]phenyl]-2-methylimidazo[1,2-b]pyridazin-8-yl]amino]ethyl]acetamide
Purity: ≥98% (HPLC)
Potent and selective PI 4-kinase  IIIβ inhibitor

Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor

Chemical Name: N-[3-[[5-Cyclopropyl-2-[[3-(4-morpholinylmethyl)phenyl]amino]-4-pyrimidinyl]amino]propyl]cyclobutanecarboxamide dihydrochloride
Purity: ≥98% (HPLC)
Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor

Potent and selective Cdc7 inhibitor

Alternate Names: BMS 863233
Chemical Name: 8-Chloro-2-(2S)-2-pyrrolidinylbenzofuro[3,2-d]pyrimidin-4(3H)-one hydrochloride
Purity: ≥98% (HPLC)
Potent and selective Cdc7 inhibitor

Potent and selective PIKfyve inhibitor

Chemical Name: 4-(6-(2-(3-Methylbenzylidene)hydrazinyl)-2-(2-(pyridin-2-yl)ethoxy)pyrimidin-4-yl)morpholine dimethanesulfonate
Purity: ≥98% (HPLC)
Potent and selective PIKfyve inhibitor

TGF-β-activated kinase (TAK1) inhibitor

Chemical Name: N-[4-[(4-Ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)benzamide
Purity: ≥98% (HPLC)
TGF-β-activated kinase (TAK1) inhibitor

Lysine deficient protein kinase (WNK) signaling inhibitor

Chemical Name: 7-Ethoxy-N3-(2-furanylmethyl)-3,9-acridinediamine
Purity: ≥98% (HPLC)
Lysine deficient protein kinase (WNK) signaling inhibitor

High affinity cyclin G associated kinase (GAK) inhibitor

Chemical Name: 6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine
Purity: ≥98% (HPLC)
High affinity cyclin G associated kinase (GAK) inhibitor

Potent TAOK inhibitor

Chemical Name: N-(2-Oxo-2-((1,2,3,4-tetrahydronaphthalen-1-yl)amino)ethyl)-[1,1'-biphenyl]-4-carboxamide
Purity: ≥98% (HPLC)
Potent TAOK inhibitor

Potent and selective LATS inhibitor; activates YAP signaling

Chemical Name: N-[4-[(3R)-Piperidin-3-yl]oxyphenyl]-1H-pyrrolo[2,3-b]pyridin-4-amine
Purity: ≥98% (HPLC)
Potent and selective LATS inhibitor; activates YAP signaling

Potent and selective MST3 kinase binding inhibitor

Chemical Name: 8-(4-Aminobutyl)-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(1,3-dihydroxypropan-2-ylamino)pyrido[2,3-d]pyrimidin-7-one trihydrochloride
Purity: ≥98% (HPLC)
Potent and selective MST3 kinase binding inhibitor

PKR inhibitor

Chemical Name: 6,8-Dihydro-8-(1H-imidazol-5-ylmethylene)-7H-pyrrolo[2,3-g]benzothiazol-7-one
Purity: ≥98% (HPLC)
PKR inhibitor

Mitochondrial pyruvate dehydrogenase kinase (PDK) inhibitor

Chemical Name: Sodium dichloroacetate
Mitochondrial pyruvate dehydrogenase kinase (PDK) inhibitor

PGK1 inhibitor; activates Nrf2

Chemical Name: (3R,4S)-rel-4-[(4-Chlorophenyl)sulfonyl]tetrahydro-N-(2-methylpropyl)-3-thiophenamine-1,1-dioxide
Purity: ≥98% (HPLC)
PGK1 inhibitor; activates Nrf2

Potent and selective pyruvate dehydrogenase kinase (PDK) 1/2/3/4 inhibitor

Chemical Name: N-[4-(2-Chloro-5-methyl-4-pyrimidinyl)phenyl]-N-[[4-[[(2,2-difluoroacetyl)amino]methyl]phenyl]methyl]-2,4-dihydroxybenzamide
Purity: ≥98% (HPLC)
Potent and selective pyruvate dehydrogenase kinase (PDK) 1/2/3/4 inhibitor

Potent and selective MST1/2 inhibitor; orally bioavailable

Chemical Name: 4-[(6,10-Dihydro-5,10-dimethyl-6-oxo-5H-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide
Purity: ≥98% (HPLC)
Potent and selective MST1/2 inhibitor; orally bioavailable

Potent and selective PIP5K1C inhibitor; antinociceptive

Chemical Name: 5-[(Cyclohexylcarbonyl)amino]-2-(phenylamino)-thiazolecarboxamide
Purity: ≥98% (HPLC)
Potent and selective PIP5K1C inhibitor; antinociceptive

Potent inhibitor of salt-inducible kinases

Chemical Name: 3-(2,4-Dimethoxyphenyl)-4-(3-thienyl)-1H-pyrrolo[2,3-b]pyridine
Purity: ≥98% (HPLC)
Potent inhibitor of salt-inducible kinases
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