Skip to main content

41 results for "Other Kinase Inhibitors" in Products

Other Kinase Inhibitors

CaM kinase III (eEF-2 kinase) inhibitor

Chemical Name:
1-Hexadecyl-2-methyl-3-(phenylmethyl)-1H-imidazolium iodide
CaM kinase III (eEF-2 kinase) inhibitor

STK33 inhibitor

Chemical Name:
N-[2-(3,4-Dihydro-3-oxo-2-quinoxalinyl)-4-(1-methylethyl)phenyl]-2-thiophenecarboxamide
Purity:
≥98%
STK33 inhibitor

Potent pan-salt inducible kinases (SIK1, SIK2 and SIK3) inhibitor. Also inhibits Lat-B-induced EP differentiation via nuclear YAP1 accumulation.

Alternate Names:
SIK inhibitor 1
Chemical Name:
1-(2,4-Dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-(6-((4-(4-methylpiperazin-1-yl)phenyl)amino)pyrimidin-4-yl)urea
Purity:
≥98%
Potent pan-salt inducible kinases (SIK1, SIK2 and SIK3) inhibitor. Also inhibits Lat-B-induced EP differentiation via nuclear YAP1 accumulation.

Potent and selective PIP5K1C inhibitor; antinociceptive

Chemical Name:
5-[(Cyclohexylcarbonyl)amino]-2-(phenylamino)-thiazolecarboxamide
Purity:
≥98%
Potent and selective PIP5K1C inhibitor; antinociceptive

Potent and selective TAK1 MAPKKK inhibitor

Chemical Name:
(3S,5Z,8S,9S,11E)-3,4,9,10-tetrahydro-8,9,16-trihydroxy-14-methoxy-3-methyl-1H-2-benzoxacyclotetradecin-1,7(8H)-dione
Purity:
≥98%
Potent and selective TAK1 MAPKKK inhibitor

Serum- and glucocorticoid-regulated kinase (SGK) inhibitor

Chemical Name:
2-Cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl-benzoic acid
Purity:
≥97%
Serum- and glucocorticoid-regulated kinase (SGK) inhibitor

Potent MSK1 inhibitor; also inhibits other AGC group kinases

Chemical Name:
2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-N-4-piperidinyl-1H-imidazo[4,5-c]pyridine-7-methanamine dihydrochloride
Purity:
≥98%
Potent MSK1 inhibitor; also inhibits other AGC group kinases

Potent and selective Tpl2 (Cot; MAP3K8) inhibitor

Chemical Name:
4-[(3-Chloro-4-fluorophenyl)amino]-6-[(3-pyridinylmethyl)amino]-1,7-naphthyridine-3-carbonitrile
Purity:
≥98%
Potent and selective Tpl2 (Cot; MAP3K8) inhibitor

Potent and selective inhibitor of Chk1 and Wee1

Chemical Name:
9-Hydroxy-4-phenyl-pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione
Purity:
≥98%
Potent and selective inhibitor of Chk1 and Wee1

Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor

Chemical Name:
4a,7a-Dihydro-2-(1-hydroxyundecyl)-1-[(4-nitrophenyl)amino]-6-phenyl-1H-pyrrolo[3,4-b]pyridine-5,7(2H,6H)-dione
Purity:
≥98%
Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor

Potent and selective Cdc7 inhibitor

Alternate Names:
BMS 863233
Chemical Name:
8-Chloro-2-(2S)-2-pyrrolidinylbenzofuro[3,2-d]pyrimidin-4(3H)-one hydrochloride
Purity:
≥98%
Potent and selective Cdc7 inhibitor

Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable

Chemical Name:
5,11-Dihydro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-11-methyl-5-(2,2,2-trifluoroethyl)-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one
Purity:
≥98%
Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable

Mitochondrial pyruvate dehydrogenase kinase (PDK) inhibitor

Chemical Name:
Sodium dichloroacetate
Mitochondrial pyruvate dehydrogenase kinase (PDK) inhibitor

Potent and selective Lck and Src inhibitor; also inhibits SIK

Alternate Names:
KIN112
Chemical Name:
2,6-Dimethylphenyl-N-(2,4-dimethoxyphenyl)-N-[2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]carbamate
Purity:
≥98%
Potent and selective Lck and Src inhibitor; also inhibits SIK

AAK1 and BMP2K inhibitor; activates Wnt signaling

Chemical Name:
N-(6-(3-((N,N-diethylsulfamoyl)amino)phenyl)-1H-indazol-3-yl)cyclopropanecarboxamide
Purity:
≥98%
AAK1 and BMP2K inhibitor; activates Wnt signaling

α1 antagonist; PGK1 activator

Chemical Name:
1-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-4-[(tetrahydro-2-furanyl)carbonyl]-piperazine hydrochloride
Purity:
≥98%
α1 and α2B antagonist (α1 > α2B). Orally active

Potent, selective and reversible CerK inhibitor

Chemical Name:
N-[2-(Benzoylamino)-6-benzothiazolyl]tricyclo[3.3.1.13,7]decane-1-carboxamide
Purity:
≥98%
Potent, selective and reversible CerK inhibitor

Dual FAK/PYK2 inhibitor

Chemical Name:
N-Methyl-N-[2-[[[2-[(2,3-dihydro-2-oxo-1H-indol-5-yl)amino]-5-(trifluoromethyl)-4-pyrimidinyl]amino]methyl]phenyl]methanesulfonamide
Purity:
≥98%
Dual FAK/PYK2 inhibitor

Potent and selective inhibitor of DAPK1

Chemical Name:
(4Z)-2-[(E)-2-Phenylethenyl)-4-(3-pyridinylmethylene)-5(4H)-oxazolone
Purity:
≥98%
Potent and selective inhibitor of DAPK1

Potent TBK inhibitor

Chemical Name:
N-[3-[[5-Cyclopropyl-2-[[4-(4-morpholinyl)phenyl]amino]-4-pyrimidinyl]amino]propyl]cyclobutanecarboxamide hydrochloride
Purity:
≥98%
Potent TBK inhibitor

PKR inhibitor

Chemical Name:
6,8-Dihydro-8-(1H-imidazol-5-ylmethylene)-7H-pyrrolo[2,3-g]benzothiazol-7-one
Purity:
≥98%
PKR inhibitor

TGF-β-activated kinase (TAK1) inhibitor

Chemical Name:
N-[4-[(4-Ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)benzamide
Purity:
≥98%
TGF-β-activated kinase (TAK1) inhibitor

Potent and selective PI 4-kinase IIIβ inhibitor

Chemical Name:
N-[2-[[6-Chloro-3-[3-[(dimethylamino)sulfonyl]phenyl]-2-methylimidazo[1,2-b]pyridazin-8-yl]amino]ethyl]acetamide
Purity:
≥98%
Potent and selective PI 4-kinase IIIβ inhibitor

Lysine deficient protein kinase (WNK) signaling inhibitor

Chemical Name:
7-Ethoxy-N3-(2-furanylmethyl)-3,9-acridinediamine
Purity:
≥98%
Lysine deficient protein kinase (WNK) signaling inhibitor

ULK inhibitor

Chemical Name:
N-[3-[[5-Cyclopropyl-2-[(1,2,3,4-tetrahydro-2-methyl-6-isoquinolinyl)amino]-4-pyrimidinyl]amino]propyl]cyclobutanecarboxamide dihydrochloride
Purity:
≥98%
ULK inhibitor
Results Per Page
5 10 25 50