Other Kinase Inhibitors: Small Molecules and Peptides
40 results for "Other Kinase Inhibitors Small Molecules and Peptides" in Products
40 results for "Other Kinase Inhibitors Small Molecules and Peptides" in Products
Other Kinase Inhibitors: Small Molecules and Peptides
Potent and selective TAK1/MAP3K7 kinase inhibitor
| Chemical Name: | N1-(1-Propyl-1H-benzimidazol-2-yl)-1,3-benzenedicarboxamide |
| Purity: | ≥98% (HPLC) |
CaM kinase III (eEF-2 kinase) inhibitor
| Chemical Name: | 1-Hexadecyl-2-methyl-3-(phenylmethyl)-1H-imidazolium iodide |
Potent and selective TAK1 MAPKKK inhibitor
| Chemical Name: | (3S,5Z,8S,9S,11E)-3,4,9,10-tetrahydro-8,9,16-trihydroxy-14-methoxy-3-methyl-1H-2-benzoxacyclotetradecin-1,7(8H)-dione |
| Purity: | ≥98% (HPLC) |
Serum- and glucocorticoid-regulated kinase (SGK) inhibitor
| Chemical Name: | 2-Cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl-benzoic acid |
| Purity: | ≥97% (HPLC) |
Potent MSK1 inhibitor; also inhibits other AGC group kinases
| Chemical Name: | 2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-N-4-piperidinyl-1H-imidazo[4,5-c]pyridine-7-methanamine dihydrochloride |
| Purity: | ≥98% (HPLC) |
Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable
| Chemical Name: | 5,11-Dihydro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-11-methyl-5-(2,2,2-trifluoroethyl)-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one |
| Purity: | ≥98% (HPLC) |
Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor
| Chemical Name: | N-[3-[[5-Cyclopropyl-2-[[3-(4-morpholinylmethyl)phenyl]amino]-4-pyrimidinyl]amino]propyl]cyclobutanecarboxamide dihydrochloride |
| Purity: | ≥98% (HPLC) |
Mitochondrial pyruvate dehydrogenase kinase (PDK) inhibitor
| Chemical Name: | Sodium dichloroacetate |
Potent and selective MST1/2 inhibitor; orally bioavailable
| Chemical Name: | 4-[(6,10-Dihydro-5,10-dimethyl-6-oxo-5H-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide |
| Purity: | ≥98% (HPLC) |
Potent and selective pyruvate dehydrogenase kinase (PDK) 1/2/3/4 inhibitor
| Chemical Name: | N-[4-(2-Chloro-5-methyl-4-pyrimidinyl)phenyl]-N-[[4-[[(2,2-difluoroacetyl)amino]methyl]phenyl]methyl]-2,4-dihydroxybenzamide |
| Purity: | ≥98% (HPLC) |
Potent and selective polynucleotide kinase/phosphatase (PNKP) inhibitor
| Chemical Name: | 4a,7a-Dihydro-2-(1-hydroxyundecyl)-1-[(4-nitrophenyl)amino]-6-phenyl-1H-pyrrolo[3,4-b]pyridine-5,7(2H,6H)-dione |
| Purity: | ≥98% (HPLC) |
Lysine deficient protein kinase (WNK) signaling inhibitor
| Chemical Name: | 7-Ethoxy-N3-(2-furanylmethyl)-3,9-acridinediamine |
| Purity: | ≥98% (HPLC) |
Potent and selective Cdc7 inhibitor
| Alternate Names: | BMS 863233 |
| Chemical Name: | 8-Chloro-2-(2S)-2-pyrrolidinylbenzofuro[3,2-d]pyrimidin-4(3H)-one hydrochloride |
| Purity: | ≥98% (HPLC) |
Potent and selective Lck and Src inhibitor; also inhibits SIK
| Alternate Names: | KIN112 |
| Chemical Name: | 2,6-Dimethylphenyl-N-(2,4-dimethoxyphenyl)-N-[2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]carbamate |
| Purity: | ≥98% (HPLC) |
Potent and selective MST3 kinase binding inhibitor
| Chemical Name: | 8-(4-Aminobutyl)-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(1,3-dihydroxypropan-2-ylamino)pyrido[2,3-d]pyrimidin-7-one trihydrochloride |
| Purity: | ≥98% (HPLC) |
Potent and selective Tpl2 (Cot; MAP3K8) inhibitor
| Chemical Name: | 4-[(3-Chloro-4-fluorophenyl)amino]-6-[(3-pyridinylmethyl)amino]-1,7-naphthyridine-3-carbonitrile |
| Purity: | ≥98% (HPLC) |
TGF-β-activated kinase (TAK1) inhibitor
| Chemical Name: | N-[4-[(4-Ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)benzamide |
| Purity: | ≥98% (HPLC) |
Potent and selective PI 4-kinase IIIβ inhibitor
| Chemical Name: | N-[2-[[6-Chloro-3-[3-[(dimethylamino)sulfonyl]phenyl]-2-methylimidazo[1,2-b]pyridazin-8-yl]amino]ethyl]acetamide |
| Purity: | ≥98% (HPLC) |
Potent pan-salt inducible kinases (SIK1, SIK2 and SIK3) inhibitor. Also inhibits Lat-B-induced EP differentiation via nuclear YAP1 accumulation.
| Alternate Names: | SIK inhibitor 1 |
| Chemical Name: | 1-(2,4-Dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-(6-((4-(4-methylpiperazin-1-yl)phenyl)amino)pyrimidin-4-yl)urea |
| Purity: | ≥98% (HPLC) |
Potent TAOK inhibitor
| Chemical Name: | N-(2-Oxo-2-((1,2,3,4-tetrahydronaphthalen-1-yl)amino)ethyl)-[1,1'-biphenyl]-4-carboxamide |
| Purity: | ≥98% (HPLC) |
PKR inhibitor
| Chemical Name: | 6,8-Dihydro-8-(1H-imidazol-5-ylmethylene)-7H-pyrrolo[2,3-g]benzothiazol-7-one |
| Purity: | ≥98% (HPLC) |
Potent and selective inhibitor of Chk1 and Wee1
| Chemical Name: | 9-Hydroxy-4-phenyl-pyrrolo[3,4-c]carbazole-1,3(2H,6H)-dione |
| Purity: | ≥98% (HPLC) |
Potent inhibitor of salt-inducible kinases
| Chemical Name: | 3-(2,4-Dimethoxyphenyl)-4-(3-thienyl)-1H-pyrrolo[2,3-b]pyridine |
| Purity: | ≥98% (HPLC) |
High affinity cyclin G associated kinase (GAK) inhibitor
| Chemical Name: | 6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine |
| Purity: | ≥98% (HPLC) |
Potent and selective LATS inhibitor; activates YAP signaling
| Chemical Name: | N-[4-[(3R)-Piperidin-3-yl]oxyphenyl]-1H-pyrrolo[2,3-b]pyridin-4-amine |
| Purity: | ≥98% (HPLC) |
