17 results for "Adenosine A2aR Small Molecules and Peptides" in Products
Adenosine A2aR Small Molecules and Peptides
Adenosine A2A Receptor (ADORA2A, Adenosine A2aR) is one of several receptor subtypes for adenosine. The activity of Adenosine A2aR, a G protein-coupled receptor family member, is mediated by G proteins which activate adenylyl cyclase. Adenosine A2aR is abundant in basal ganglia, vasculature and platelets and is a major target of caffeine. Variability in the acute blood pressure response to coffee may be partly explained by genetic polymorphisms of the adenosine A2A receptors, including Adenosine A2aR, and alpha(2)-adrenergic receptors.
A2A agonist
Potent and highly selective A2A antagonist
Potent, highly selective A2A antagonist
High affinity adenosine agonist
Very selective, high affinity A2A antagonist
Endogenous adenosine receptor agonist
A1 and A2B antagonist. CNS stimulant
PDE inhibitor (non-selective)
Adenosine receptor agonist
Potent adenosine A2A agonist
Potent adenosine receptor antagonist
Adenosine A2A antagonist
Adenosine receptor antagonist
Potent adenosine A2A and A2B receptor partial agonist
Potent and selective A2A antagonist
Selective A2B antagonist
Potent and selective A2A antagonist
