47 results for "Bromodomain Inhibitors" in Products

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Bromodomain Inhibitors

(+)-JQ1
Catalog #: 4499
(2)
Citations (46)
Product Documents
Images (1)

Potent and selective BET bromodomain inhibitor; cell permeable

Chemical Name:
(6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid 1,1-dimethylethyl ester
Purity:
≥98%
Potent and selective BET bromodomain inhibitor; cell permeable
Catalog #
Availability
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Qty
4499/10
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MZ 1
Catalog #: 6154
Citations (19)
Product Documents
Images (2)

(+)-JQ1 based Degrader (PROTAC®) that preferentially degrades BRD4

Chemical Name:
(2S,4R)-1-((S)-2-(tert-butyl)-17-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,16-dioxo-6,9,12-trioxa-3,15-diazaheptadecanoyl)- 4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity:
≥98%
Application of MZ 1 in HeLa Cells
(2)
Catalog #
Availability
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Qty
6154/5
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I-BET 151 dihydrochloride
Catalog #: 4650
(2)
Citations (10)
Product Documents
Images (1)

BET bromodomain inhibitor; also promotes differentiation of hiPSCs into megakaryocytes

Chemical Name:
7-(3,5-Dimethyl-4-isoxazolyl)-1,3-dihydroxy-8-methoxy-1-[(1R)-1-(2-pyridinyl)ethyl]-2H-imidazo[4,5-c]quinolin-2-one dihydrochloride
Purity:
≥98%
BET bromodomain inhibitor; also promotes differentiation of hiPSCs into megakaryocytes
Catalog #
Availability
Size / Price
Qty
4650/10
4650/50
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dBRD9
Catalog #: 6606
Citations (12)
Product Documents
Images (1)

Potent and selective BRD9 Degrader (PROTAC®)

Chemical Name:
2-[[[4-(1,2-Dihydro-2-methyl-1-oxo-2,7-naphthyridin-4-yl)-2-6-dimethoxyphenyl]methyl]methylamino]-N-[2-[2-[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]amino]ethoxy]ethoxy]ethyl]acetamide dihydrochloride
Purity:
≥98%
Potent and selective BRD9 Degrader (PROTAC®)
Catalog #
Availability
Size / Price
Qty
6606/5
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XMD 8-92
Catalog #: 4132
Citations (13)
Product Documents
Images (1)

ERK5/BMK1 inhibitor; also BRD4 inhibitor

Chemical Name:
2-[[2-Ethoxy-4-(4-hydroxy-1-piperidinyl)phenyl]amino]-5,11-dihydro-5,11-dimethyl-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one
Purity:
≥98%
ERK5/BMK1 inhibitor; also BRD4 inhibitor
Catalog #
Availability
Size / Price
Qty
4132/50
4132/10
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I-BRD9
Catalog #: 5591
Citations (11)
Product Documents
Images (1)

Potent and selective BRD9 inhibitor

Chemical Name:
5-Ethyl-4,5-dihydro-4-oxo-N-(tetrahydro-1,1-dioxido-2H-thiopyran-4-yl)-7-[3-(trifluoromethyl)phenyl]thieno[3,2-c]pyridine-2-carboximidamide
Purity:
≥98%
Potent and selective BRD9 inhibitor
Catalog #
Availability
Size / Price
Qty
5591/50
5591/10
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cis MZ 1
Catalog #: 6155
Citations (1)
Product Documents
Images (1)

Negative Control for MZ 1 (Cat. No. 6154)

Chemical Name:
(2S,4S)-1-((S)-2-(tert-butyl)-17-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,16-dioxo-6,9,12-trioxa-3,15-diazaheptadecanoyl)- 4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity:
≥98%
Negative Control for MZ 1 (Cat. No. 6154)
Catalog #
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Qty
6155/5
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dBET1
Catalog #: 6327
Citations (4)
Product Documents
Images (1)

(+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo

Chemical Name:
(6S)-4-(4-Chlorophenyl)-N-[4-[[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]acetyl]amino]butyl]-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide
Purity:
≥98%
(+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo
Catalog #
Availability
Size / Price
Qty
6327/5
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dBRD9-A
Catalog #: 6943
Citations (5)
Product Documents
Images (1)

Potent BRD9 Degrader (PROTAC®)

Chemical Name:
2-((2,6-Dimethoxy-4-(2-methyl-1-oxo-1,2-dihydro-2,7-naphthyridin-4-yl)benzyl)(methyl)amino)-N-(8-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)octyl)acetamide
Purity:
≥98%
Potent BRD9 Degrader (PROTAC®)
Catalog #
Availability
Size / Price
Qty
6943/5
Bulk Order

dBET6
Catalog #: 6945
Citations (8)
Product Documents
Images (1)

Potent and selective (+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo

Chemical Name:
(6S)-4-(4-Chlorophenyl)-N-[8-[[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]acetyl]amino]octyl]-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide
Purity:
≥98%
Potent and selective (+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo
Catalog #
Availability
Size / Price
Qty
6945/5
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PFI 1
Catalog #: 4445
Citations (5)
Product Documents
Images (1)

BET bromodomain inhibitor

Chemical Name:
2-Methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide
Purity:
≥98%
BET bromodomain inhibitor
Catalog #
Availability
Size / Price
Qty
4445/10
4445/50
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Bromosporine
Catalog #: 4758
Citations (3)
Product Documents
Images (1)

Broad spectrum bromodomain inhibitor

Chemical Name:
N-[(6-3-Methanesulfonamido-4-methylphenyl)-3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-8-yl]carbamate
Purity:
≥98%
Broad spectrum bromodomain inhibitor
Catalog #
Availability
Size / Price
Qty
4758/10
Bulk Order

SGC-CBP30
Catalog #: 4889
(1)
Citations (13)
Product Documents
Images (1)

Potent CBP/p300 BRD inhibitor

Chemical Name:
2-[2-(3-Chloro-4-methoxyphenyl)ethyl]-5-(dimethyl-1,2-oxazol-4-yl)-1-[(2S)-2-(morpholin-4-yl)propyl]-1H-1,3-benzodiazole
Purity:
≥98%
Potent CBP/p300 BRD inhibitor
Catalog #
Availability
Size / Price
Qty
4889/50
4889/10
Bulk Order

PFI 3
Catalog #: 5072
Citations (7)
Product Documents
Images (1)

Potent and selective SMARCA2/4 and polybromo 1 inhibitor

Chemical Name:
(2E)-1-(2-Hydroxyphenyl)-3-[(1R,4R)-5-(pyridin-2-yl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]prop-2-en-1-one
Purity:
≥98%
Potent and selective SMARCA2/4 and polybromo 1 inhibitor
Catalog #
Availability
Size / Price
Qty
5072/10
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BAZ2-ICR
Catalog #: 5266
Citations (2)
Product Documents
Images (1)

Selective BAZ2 inhibitor

Chemical Name:
4-[4-(1-Methyl-1H-pyrazole-4-yl)-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-5-yl]benzonitrile
Purity:
≥98%
Selective BAZ2 inhibitor
Catalog #
Availability
Size / Price
Qty
5266/50
5266/10
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CPI 203
Catalog #: 5331
(1)
Citations (3)
Product Documents
Images (1)

BET bromodomain inhibitor; arrests cell cycle at G1 phase

Alternate Names:
TEN 010
Chemical Name:
(6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide
Purity:
≥98%
BET bromodomain inhibitor; arrests cell cycle at G1 phase
Catalog #
Availability
Size / Price
Qty
5331/10
Bulk Order

NI 57
Catalog #: 5546
Citations (1)
Product Documents
Images (1)

Potent and selective BRPF bromodomain inhibitor

Chemical Name:
4-Cyano-N-(1,3-dimethyl-2-oxo-1,2-dihydroquinolin-6-yl)-2-methoxybenzene-1-sulfonamide
Purity:
≥98%
Potent and selective BRPF bromodomain inhibitor
Catalog #
Availability
Size / Price
Qty
5546/50
5546/10
Bulk Order

BI 9564
Catalog #: 5590
Citations (6)
Product Documents
Images (1)

Potent and selective BRD9 and BRD7 inhibitor; orally active

Chemical Name:
4-[4-[(Dimethylamino)methyl]-2,5-dimethoxyphenyl]-2-methyl-1,2-dihydro-2,7-naphthyridin-1-one
Purity:
≥98%
Potent and selective BRD9 and BRD7 inhibitor; orally active
Catalog #
Availability
Size / Price
Qty
5590/10
Bulk Order

(-)-JQ1
Catalog #: 5603
Citations (74)
Product Documents
Images (1)

Negative control for (+)-JQ1

Chemical Name:
(6R)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid 1,1-dimethylethyl ester
Purity:
≥98%
Negative control for (+)-JQ1
Catalog #
Availability
Size / Price
Qty
5603/10
Bulk Order

LP 99
Catalog #: 5496
Product Documents
Images (1)

Selective BRD7 and BRD9 inhibitor

Chemical Name:
N-[(2R,3S)-2-(4-Chlorophenyl)-1-(1,2-dihydro-1,4-dimethyl-2-oxo-7-quinolinyl)-6-oxo-3-piperidinyl]-2-methyl-1-propanesulfonamide
Purity:
≥98%
Selective BRD7 and BRD9 inhibitor
Catalog #
Availability
Size / Price
Qty
5496/5
5496/25
Bulk Order

ent-LP 99
Catalog #: 5497
Product Documents
Images (1)

Negative Control for LP 99

Chemical Name:
N-[(2S,3R)-2-(4-Chlorophenyl)-1-(1,2-dihydro-1,4-dimethyl-2-oxo-7-quinolinyl)-6-oxo-3-piperidinyl]-2-methyl-1-propanesulfonamide
Purity:
≥98%
Negative Control for LP 99
Catalog #
Availability
Size / Price
Qty
5497/5
5497/25
Bulk Order

NVS-CECR2-1
Catalog #: 5744
Citations (2)
Product Documents
Images (1)

Potent and selective CECR2 inhibitor

Chemical Name:
N-Cyclopropyl-2-(propylsulfonyl)-6-(1-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-indol-5-yl)pyrimidin-4-amine
Purity:
≥98%
Potent and selective CECR2 inhibitor
Catalog #
Availability
Size / Price
Qty
5744/50
5744/10
Bulk Order

BAY 299
Catalog #: 5970
Citations (2)
Product Documents
Images (1)

Potent and selective BRD1 and TAF1 inhibitor

Chemical Name:
6-(3-Hydroxypropyl)-2-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)-1H-benzo[de]isoquinoline-1,3(2H)-dione
Purity:
≥98%
Potent and selective BRD1 and TAF1 inhibitor
Catalog #
Availability
Size / Price
Qty
5970/25
5970/5
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TP 472N
Catalog #: 5999
Citations (1)
Product Documents
Images (1)

Negative control for TP 472

Chemical Name:
1-(8-(2-(Cyclopropylmethoxy)phenyl)pyrrolo[1,2-a]pyrimidin-6-yl)ethanone
Purity:
≥98%
Negative control for TP 472
Catalog #
Availability
Size / Price
Qty
5999/10
Bulk Order

TP 472
Catalog #: 6000
Citations (57)
Product Documents
Images (1)

Potent BRD9/7 inhibitor

Chemical Name:
3-(6-Acetylpyrrolo[1,2-a]pyrimidin-8-yl)-N-cyclopropyl-4-methylbenzamide
Purity:
≥98%
Potent BRD9/7 inhibitor
Catalog #
Availability
Size / Price
Qty
6000/10
Bulk Order
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