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GABA-B Receptor Antagonists: Small Molecules and Peptides

GABAB receptors are metabotropic G-protein-coupled receptors (GPCRs). They are responsible for mediating the inhibitory effects of GABA and ionotropic GABAA and GABAA-ρ receptors.

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8 results for "GABA-B Receptor Antagonists Small Molecules and Peptides" in Products

8 results for "GABA-B Receptor Antagonists Small Molecules and Peptides" in Products

GABA-B Receptor Antagonists: Small Molecules and Peptides

GABAB receptors are metabotropic G-protein-coupled receptors (GPCRs). They are responsible for mediating the inhibitory effects of GABA and ionotropic GABAA and GABAA-ρ receptors.

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Potent and selective GABAB antagonist

Chemical Name: (2S)-3-[[(1S)-1-(3,4-Dichlorophenyl)ethyl]amino-2-hydroxypropyl](phenylmethyl)phosphinic acid hydrochloride
Purity: ≥98% (HPLC)
Potent and selective GABAB antagonist

Selective GABAB antagonist; brain penetrant

Chemical Name: (3-Aminopropyl)(diethoxymethyl)phosphinic acid
Selective GABAB antagonist; brain penetrant

Selective and competitive GABAB antagonist; orally bioavailable

Chemical Name: (2S)-(+)-5,5-Dimethyl-2-morpholineacetic acid
Purity: ≥98%
Selective and competitive GABAB antagonist; orally bioavailable

GABAB antagonist; displays activity at presynaptic receptors

Chemical Name: (3-Aminopropyl)ethylphosphinic acid hydrochloride
Purity: ≥98% (HPLC)
GABAB antagonist; displays activity at presynaptic receptors

Potent and selective GABAB antagonist

Chemical Name: [S-(R*,R*)]-[3-[[1-(3,4-Dichlorophenyl)ethyl]amino]-2-hydroxypropyl](cyclohexylmethyl) phosphinic acid
Purity: ≥96% (HPLC)
Potent and selective GABAB antagonist

Selective GABAB antagonist

Chemical Name: (RS)-3-Amino-2-(4-chlorophenyl)propylsulfonic acid
Purity: ≥98% (HPLC)
Selective GABAB antagonist

Potent and selective GABAB antagonist

Chemical Name: 3-[[(3,4-Dichlorophenyl)methyl]amino]propyl] diethoxymethyl)phosphinic acid
Purity: ≥98% (HPLC)
Potent and selective GABAB antagonist

Selective GABAB antagonist; more potent than Saclofen (Cat. No. 0246)

Chemical Name: (RS)-3-Amino-2-(4-chlorophenyl)-2-hydroxypropyl-sulfonic acid
Selective GABAB antagonist; more potent than Saclofen (Cat. No. 0246)
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