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10 results for "Casein Kinase 1 Inhibitors" in Products

Casein Kinase 1 Inhibitors

Potent p38 MAPK inhibitor; anti-inflammatory

Chemical Name:
N-[4-[2-Ethyl-4-(3-methylphenyl)-5-thiazolyl]-2-pyridinyl]benzamide
Purity:
≥98%
Potent p38 MAPK inhibitor; anti-inflammatory

CK1 inhibitor

Chemical Name:
N-(2-Aminoethyl)-5-chloro-8-isoquinolinesulfonamide dihydrochloride
Purity:
≥99%
CK1 inhibitor

Cdk inhibitor; potently inhibits cdk1 and cdk2; also inhibits CK1; acts as molecular glue

Chemical Name:
(2R)-2-[[9-(Methylethyl)-6-[[[4-(2-pyridinyl)phenyl]methyl]amino]-9H-purin-2-yl]amino]-1-butanol trihydrochloride
Purity:
≥98%
Cdk inhibitor; potently inhibits cdk1 and cdk2; also inhibits CK1; acts as molecular glue

Potent and selective CK1ε and CK1δ inhibitor

Chemical Name:
4-[1-Cyclohexyl-4-(4-fluorophenyl)-1H-imidazol-5-yl]-2-pyrimidinamine dihydrochloride
Purity:
≥98%
Potent and selective CK1ε and CK1δ inhibitor

Selective CK1 inhibitor. Also inhibits TGF-βRI

Chemical Name:
4-[4-(2,3-Dihydro-1,4-benzodioxin-6-yl)-5-(2-pyridinyl)-1H-imidazol-2-yl]benzamide
Purity:
≥98%
Selective CK1 inhibitor. Also inhibits TGF-βRI

Selective casein kinase 1ε inhibitor

Chemical Name:
3-[(3-Chlorophenoxy)methyl]-1-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine hydrochloride
Purity:
≥98%
Selective casein kinase 1ε inhibitor

Potent CK1 inhibitor; also inhibits cyclin-dependent kinases

Chemical Name:
2-[[9-(1-Methylethyl)-6-[[3-(2-pyridinyl)phenyl]amino]-9H-purin-2-yl]amino]-1-butanol dihydrochloride
Purity:
≥98%
Potent CK1 inhibitor; also inhibits cyclin-dependent kinases

Potent CK1δ/ε inhibitor

Chemical Name:
4-[4-(4-Fluorophenyl)-1-[1-(3-isoxazolylmethyl)-4-piperidinyl]-1H-imidazol-5-yl]-2-pyrimidinamine
Purity:
≥98%
Potent CK1δ/ε inhibitor

Potent and selective CK1α, CK1δ and CK1ε inhibitor

Chemical Name:
4-(1-((4-Fluoro-1-methylpiperidin-4-yl)methyl)-4-(5-fluoropyridin-2-yl)-1H-imidazol-5-yl)-1H-pyrrolo[2,3-b]pyridine
Purity:
≥98%
Potent and selective CK1α, CK1δ and CK1ε inhibitor

Potent and selective CK1α molecular glue Degrader

Chemical Name:
3-(5-(Benzo[d]isoxazol-3-ylamino)-1-oxoisoindolin-2-yl)piperidine-2,6-dione
Purity:
≥98%
Potent and selective CK1α molecular glue Degrader
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