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23 results for "voltage-gated-sodium-channel-blockers&view=expanded" in Products

Na+ channel blocker

Alternate Names:
TTx
Chemical Name:
(4R,4aR,5R,7S,9S,10S,10aR,11S,12S)-Octahydro-12-(hydroxymethyl)-2-imino-5,9:7,10a-dimethano-10aH-[1,3]dioxocino[6,5-d]pyrimidine-4,7,10,11,12-pentol
Purity:
≥98%
Na+ channel blocker

Na+ channel blocker

Chemical Name:
N-(2,6-Dimethylphenylcarbamoylmethyl)triethylammonium bromide
Purity:
≥98%
Na+ channel blocker

Na+ channel blocker; also I2 imidazoline ligand

Chemical Name:
3,5-Diamino-N-(aminoiminomethyl)-6-chloropyrazinecarboxamide hydrochloride
Purity:
≥98%
Na+ channel blocker; also I2 imidazoline ligand

Potent hNav1.4, rNav1.6 and rNav1.7 channel activator

Purity:
≥95%
Potent hNav1.4, rNav1.6 and rNav1.7 channel activator

Non-selective Ca2+ channel blocker; also NCX inhibitor

Chemical Name:
N-Benzyl-N-(3-isobutoxy-2-pyrrolidin-1-yl-propyl)aniline hydrochloride
Purity:
≥98%
Non-selective Ca2+ channel blocker; also NCX inhibitor

Selective NaV1.7 channel blocker

Purity:
≥95%
Selective NaV1.7 channel blocker

Potent voltage-dependent NaV1.8 channel blocker

Chemical Name:
5-(4-Butoxy-3-chlorophenyl)-N-[[2-(4-morpholinyl)-3-pyridinyl]methyl-3-pyridine carboxamide
Purity:
≥97%
Potent voltage-dependent NaV1.8 channel blocker

Cardiac Na+ channel blocker. Antiarrhythmic

Chemical Name:
N-(2-Piperidylmethyl)-2,5-bis-(2,2,2-trifluoroethoxy)benzamide acetate
Purity:
≥98%
Cardiac Na+ channel blocker. Antiarrhythmic

Na+ channel blocker

Chemical Name:
N-(2,6-Dimethylphenylcarbamoylmethyl)triethylammonium chloride
Purity:
≥98%
Na+ channel blocker

Selective NaV1.8 channel blocker

Chemical Name:
5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)-2-furancarboxamide
Purity:
≥98%
Selective NaV1.8 channel blocker
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