Calcium-sensing R/CaSR: Small Molecules and Peptides
5 results for "Calcium-sensing R/CaSR Small Molecules and Peptides" in Products
5 results for "Calcium-sensing R/CaSR Small Molecules and Peptides" in Products
Calcium-sensing R/CaSR: Small Molecules and Peptides
Positive allosteric modulator of human calcium-sensing receptor (CaSR)
| Chemical Name: | 2-Chloro-N-[(1R)-1-(3-methoxyphenyl)ethyl]-benzenepropanamine hydrochloride |
| Purity: | ≥98% (HPLC) |
Allosteric Calcium-sensing receptor (CaSR) agonist; also CYP2D2 inhibitor and Ca2+ channel blocker; orally bioavailable
| Alternate Names: | AMG 073 |
| Chemical Name: | N-[(1R)-1-(1-Naphthyl)ethyl]-3-[3-(trifluoromethyl)phenyl]propan-1-amine hydrochloride |
| Purity: | ≥98% (HPLC) |
Selective calcium-sensing receptor (CaSR) antagonist; orally active calcilytic agent
| Chemical Name: | 2-Chloro-6-[(2R)-3-[[1,1-dimethyl-2-(2-naphthalenyl)ethyl]amino-2-hydroxypropoxy]benzonitrile hydrochloride |
| Purity: | ≥98% (HPLC) |
Negative allosteric modulator of calcium-sensing receptor (CaSR)
| Chemical Name: | 4-Chloro-N-[(1S,2S)-2-[[(1R)-1-(1-naphthalenyl)ethyl]amino]cyclohexyl]-benzamide hydrochloride |
| Purity: | ≥98% (HPLC) |
Biased allosteric modulator of calcium-sensing receptor (CaSR)
| Chemical Name: | α-(2,4-Dimethylphenyl)-α-methyl-2-benzothiazolemethanol |
| Purity: | ≥98% (HPLC) |
