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21 results for "beta-catenin-inhibitors&view=expanded" in Products

PORCN inhibitor; inhibits Wnt processing and secretion

Chemical Name:
N-(6-Methyl-2-benzothiazolyl)-2-[(3,4,6,7-tetrahydro-4-oxo-3-phenylthieno[3,2-d]pyrimidin-2-yl)thio]-acetamide
Purity:
≥98%
iPSC-derived heart organoids differentiated with IWP 2 and CHIR 99021
(2)

Potent tankyrase inhibitor

GMP Version Available: TB3748-GMP
GMP
Alternate Names:
XAV939 Wnt Signaling Inhibitor
Chemical Name:
3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one
Purity:
≥98%
Potent tankyrase inhibitor

Potent p38 MAPK inhibitor; anti-inflammatory

Chemical Name:
N-[4-[2-Ethyl-4-(3-methylphenyl)-5-thiazolyl]-2-pyridinyl]benzamide
Purity:
≥98%
Potent p38 MAPK inhibitor; anti-inflammatory

Wnt/β-catenin signaling inhibitor; axin stabilizer

Chemical Name:
rel-4-[(3aR,4S,7R,7aS)-1,3,3a,4,7,7a-Hexahydro-1,3-dioxo-4,7-methano-2H-isoindol-2-yl]-N-8-quinolinylbenzamide
Purity:
≥98%
Wnt/β-catenin signaling inhibitor; axin stabilizer

Inhibits TCF/β-catenin-mediated transcription

Chemical Name:
(6S,9aS)-Hexahydro-6-[(4-hydroxyphenyl)methyl]-8-(1-naphthalenylmethyl)-4,7-dioxo-N-(phenylmethyl)-2H-pyrazino[1,2-a]pyrimidine-1(6H)-carboxamide
Purity:
≥98%
Inhibits TCF/β-catenin-mediated transcription

Wnt signaling inhibitor; inhibits β-catenin-transcription factor interactions

Purity:
≥95%
Wnt signaling inhibitor; inhibits β-catenin-transcription factor interactions

Inhibits β-catenin-responsive transcription (CRT)

Chemical Name:
5-[[2,5-Dimethyl-1-(3-pyridinyl)-1H-pyrrol-3-yl]methylene]-3-phenyl-2,4-thiazolidinedion
Purity:
≥98%
Inhibits β-catenin-responsive transcription (CRT)

Inhibitor of mutant β-catenin signaling in hepatocellular carcinoma

Chemical Name:
4-[3-Fluoro-4-[[[[4-(1,1,2,2,2-pentafluoroethyl)phenyl]amino]carbonyl]amino]phenoxy]-N-methyl-2-pyridinecarboxamide
Purity:
≥98%
Inhibitor of mutant β-catenin signaling in hepatocellular carcinoma

Potent inhibitor of Wnt/β-catenin signaling

Chemical Name:
N-(6-Methyl-2-benzothiazolyl)-2-[(3,4,6,7-tetrahydro-3-(2-methoxyphenyl)-4-oxothieno[3,2-d]pyrimidin-2-yl)thio]-acetamide
Purity:
≥98%
Potent inhibitor of Wnt/β-catenin signaling

Inhibitor of Wnt/β-catenin signaling

Chemical Name:
N-[4-(4-Ethyl-1-piperazinyl)phenyl]-2-oxo-2H-1-benzopyran-3-carboxamide
Purity:
≥98%
Inhibitor of Wnt/β-catenin signaling
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