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11 results for "Histamine H1 R Small Molecules and Peptides" in Products

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Histamine H1 R Small Molecules and Peptides

Histamine H1R (HRH1) is a G-protein coupled 7-transmembrane putative glycoprotein that is implicated in the pathogenesis of asthma and is a major pharmaceutical target for antihistamines. It has been detected as a mixture of monomers and homodimers, with highest concentration in the placenta, followed by brain, lung (produced by airway smooth muscle, bronchial epithelium and macrophages) and other tissues.

Meclizine dihydrochloride

Catalog #: 4245

Product Documents

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Human pregnane X receptor agonist; H1 antagonist

Alternate Names:

Meclozine

Chemical Name:

1-[(4-Chlorophenyl)phenylmethyl]4-[(3-methylphenyl)methyl]piperazine dihydrochloride

Purity:

≥99%

Terfenadine

Catalog #: 3948

(1)

Product Documents

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H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker

Chemical Name:

α-[4-(1,1-Dimethylethyl)phenyl]-4-(hydroxydiphenylmethyl)-1-piperidinebutanol

Purity:

≥98%

Clemastine fumarate

Catalog #: 1453

Product Documents

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H1 antagonist

Chemical Name:

(2R)-2-[2-[(1R)-1-(4-Chlorophenylethoxy]ethyl]-1-methyl-2-pyrrolidine fumarate

Purity:

≥98%

Mirtazapine

Catalog #: 2018

Citations (523)

Product Documents

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Potent 5-HT2 antagonist; also 5-HT3, H1 and α2 antagonist; antidepressant

Alternate Names:

Org 3770,6-Azamianserin

Chemical Name:

1,2,3,4,10,14b-Hexahydro-2-methylpyrazino[2,1-a]pyrido[2,3-c][2]benzazepine

Purity:

≥98%

2-Pyridylethylamine dihydrochloride

Catalog #: 2478

Product Documents

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H1 agonist

Chemical Name:

2-Pyridineethanamine dihydrochloride

Purity:

≥99%

HTMT dimaleate

Catalog #: 0646

Product Documents

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H1/ H2 agonist

Alternate Names:

Histamine trifluoromethyl toluidide

Chemical Name:

6-[2-(4-Imidazolyl)ethylamino]-N-(4-trifluoromethylphenyl)heptanecarboxamide dimaleate

Purity:

≥99%

Histamine dihydrochloride

Catalog #: 3545

(1)

Product Documents

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Endogenous histamine receptor agonist

Chemical Name:

2-(4-Imidazolyl)ethylamine dihydrochloride

Olopatadine hydrochloride

Catalog #: 4241

Product Documents

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H1 antagonist; ocular antiallergic agent

Chemical Name:

(Z)-11-[3-(Dimethylamino)propylidene]-6,11-dihydro-dibenz[b,e]oxepin-2-acetic acid hydrochloride

Purity:

≥98%

Diphenhydramine hydrochloride

Catalog #: 3072

Product Documents

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H1 antagonist

Alternate Names:

DPH

Chemical Name:

2-Diphenylmethoxy-N,N-dimethylethanamine hydrochloride

Purity:

≥98%

Astemizole

Catalog #: 3489

(1)

Product Documents

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Orally active, potent H1 antagonist; also KV11.1 (hERG) channel blocker

Alternate Names:

Hismanal

Chemical Name:

1-[(4-Fluorophenyl)methyl]-N-[1-[2-(4-methoxyphenyl)ethyl]-4-piperidinyl]-1H-benzimidazol-2-amine

Purity:

≥98%

Asenapine maleate

Catalog #: 3737

Product Documents

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Non-selective 5-HT, dopamine, adrenalin and histamine receptor antagonist; antipsychotic agent

Chemical Name:

(3aR*,12bR*)-5-Chloro-2,3,3a,12b-tetrahydro-2-methyl-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole maleate

Purity:

≥98%

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