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23 results for "egf-receptor-inhibitors&view=expanded" in Products

Highly potent EGFR-kinase inhibitor

Alternate Names:
Tyrphostin AG 1478
Chemical Name:
N-(3-Chlorophenyl)-6,7-dimethoxy-4-quinazolinanine hydrochloride
Purity:
≥98%
Highly potent EGFR-kinase inhibitor

Orally active, selective EGFR inhibitor

Alternate Names:
Gefitinib,ZD 1839
Chemical Name:
N-(3-Chloro-4-fluorophenyl)-7-methoxy-6-[3-(4-morpholinyl)propoxy]-4-quinazolinamine
Purity:
≥98%
Orally active, selective EGFR inhibitor

EGFR kinase inhibitor. Also estrogen and PPARγ ligand

Chemical Name:
5,7-Dihydroxy-3-(4-hydroxyphenyl)-4H-1-benzopyran-4-one
Purity:
≥98%
EGFR kinase inhibitor. Also estrogen and PPARγ ligand

EGFR-kinase inhibitor. Also JAK2, JAK3 inhibitor

Alternate Names:
Tyrphostin AG 490
Chemical Name:
(E)-2-Cyano-3-(3,4-dihydrophenyl)-N-(phenylmethyl)-2-propenamide
Purity:
≥98%
EGFR-kinase inhibitor. Also JAK2, JAK3 inhibitor

Potent, reversible EGFR tyrosine kinase inhibitor

Chemical Name:
N-(3-Ethynylphenyl)-6,7-bis(2-methoxyethoxy)-4-quinazolinamine hydrochloride
Purity:
≥98%
Potent, reversible EGFR tyrosine kinase inhibitor

Highly potent EGFR and ErbB2 inhibitor; inhibts wild type and mutated receptors

Chemical Name:
(4-Fluorophenyl)methyl N-[2-[(1-methyl-1H-pyrazol-4-yl)amino]-4-pyrimidinyl]-N-[3-[(1-oxo-2-propen-1-yl)amino]phenyl]carbamate
Purity:
≥98%
Highly potent EGFR and ErbB2 inhibitor; inhibts wild type and mutated receptors

Potent ErbB receptor family inhibitor

Chemical Name:
N4-(3-Bromophenyl)-N6-methyl-pyrido[3,4-d]pyrimidine-4,6-diamine
Purity:
≥98%
Potent ErbB receptor family inhibitor

Potent ErbB receptor family inhibitor

Chemical Name:
5E-4-Amino-6-(4-benzyloxy-3-chlorophenylamino)pyrimidine-5-carboxaldehyde N-(2-morpholin-4-ylethyl) oxime hydrochloride
Purity:
≥97%
Potent ErbB receptor family inhibitor

Potent dual EGFR/ErbB2 inhibitor; orally active

Chemical Name:
N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[2-[[[2-(methylsulfonyl)ethyl]amino]methyl]-4-thiazolyl]-4-quinazolinamine dihydrochloride
Purity:
≥97%
Potent dual EGFR/ErbB2 inhibitor; orally active

Potent and selective ErbB2 inhibitor

Alternate Names:
Mubritinib
Chemical Name:
1-[4-[4-[[2-[(1E)-2-[4-(trifluoromethyl)phenyl]ethenyl]-4-oxazolyl]methoxy]phenyl]butyl]-1H-1,2,3-triazole
Purity:
≥98%
Potent and selective ErbB2 inhibitor
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