3 results for "Protein Kinase D Inhibitors Small Molecules and Peptides" in Products
Protein Kinase D Inhibitors: Small Molecules and Peptides
The protein kinase D (PKD) family of serine/threonine protein kinases contains three members; PKD1, PKD2 and PKD3. These enzymes occupy a unique position in the signal transduction pathway initiated by diacylglycerol (DAG) and protein kinase C (PKC). PKDs are direct targets of DAG, and also lie downstream of PKC in a novel signal transduction pathway that is implicated in a variety of biological processes.
Structurally, PKDs contain an N' terminal cysteine-rich domain (CRD), which binds ...
Selective protein kinase D inhibitor
| Chemical Name: | 2,3,4,5-Tetrahydro-7-hydroxy-1H-benzofuro[2,3-c]azepin-1-one |
| Purity: | ≥98% (HPLC) |
Potent protein kinase D (PKD) inhibitor
| Chemical Name: | 2-[4-[[(2R)-2-aminobutyl]amino]-2-pyrimidinyl]-4-(1-methyl-1H-pyrazol-4-yl)phenol dihydrochloride |
| Purity: | ≥98% (HPLC) |
Selective PKD inhibitor; analog of CID 755673 (Cat. No. 3327)
| Chemical Name: | 9-Hydroxy-3,4-dihydro-2H-[1]-benzothiolo[2,3-f][1,4]thiazepin-5-one |
| Purity: | ≥98% (HPLC) |
