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30 results for "dehydrogenase-inhibitors&view=expanded" in Products

PDH and KGDH inhibitor

Chemical Name:
6,8-Bis[(phenylmethyl)thio]octanoic acid
Purity:
≥98%
PDH and KGDH inhibitor

ALDH1A2 inhibitor

Chemical Name:
N,N'-1,8-Octanediylbis(2,2-dichloroacetamide)
ALDH1A2 inhibitor

Potent and selective LDHA inhibitor

Chemical Name:
3-[[3-[(Cyclopropylamino)sulfonyl]-7-(2,4-dimethoxy-5-pyrimidinyl)-4-quinolinyl]amino]-5-(3,5-difluorophenoxy)benzoic acid
Purity:
≥98%
Potent and selective LDHA inhibitor

Potent and selective inhibitor of mutant isocitrate dehydrogenase 1 (mIDH1)

Chemical Name:
N-[2-(Cyclohexylamino)-1-(2-methylphenyl)-2-oxoethyl]-N-(3-fluorophenyl)-2-methyl-1H-Imidazole-1-acetamide
Purity:
≥98%
Potent and selective inhibitor of mutant isocitrate dehydrogenase 1 (mIDH1)

Potent inhibitor of mutant isocitrate dehydrogenase (mIDH1)

Chemical Name:
(2S)-N-{(1S)-1-(2-Chlorophenyl)-2-[(3,3-difluorocyclobutyl)amino]-2-oxoethyl}-1(4-cyanopyridin-2-yl)-N-(5-fluoropyridin-3-yl)-5-oxopyrrolidine-2-carboxamide
Purity:
≥98%
Potent inhibitor of mutant isocitrate dehydrogenase (mIDH1)

Potent and selective DHODH inhibitor

Alternate Names:
BRQ,DuP 785,NSC 368390
Chemical Name:
6-Fluoro-2-(2'-fluoro[1,1'-biphenyl]-4-yl)-3-methyl-4-quinolinecarboxylic acid sodium
Purity:
≥98%
Potent and selective DHODH inhibitor

Reversibly stimulates SERCA Ca2+-ATPase; displays a range of other activities

Alternate Names:
Tetraethylthiuram disulfide
Chemical Name:
Bis(diethylthiocarbamyoyl)disulfide
Reversibly stimulates SERCA Ca2+-ATPase; displays a range of other activities

Inhibitor of DHODH; active metabolite of Leflunomide

Alternate Names:
A77 1726
Chemical Name:
2-Cyano-3-hydroxy-N-[4-(trifluoromethyl)phenyl]-2-butenamide
Purity:
≥98%
Inhibitor of DHODH; active metabolite of Leflunomide

Inosine monophosphatase dehydrogenase (IMPDH) inhibitor

Chemical Name:
6-(1,3-Dihydro-4-hydroxy-6-methoxy-7-methyl-3-oxo-5-isobenzofuranyl)-4-methyl-4-hexenoic acid
Purity:
≥98%
Inosine monophosphatase dehydrogenase (IMPDH) inhibitor

Inosine monophosphatase dehydrogenase (IMPDH) inhibitor

Chemical Name:
N-[1-[6-(4-Ethyl-1-piperazinyl)-3-pyridinyl]-1-methylethyl]-2-fluoro-9,10-dihydro-9-oxo-3-acridinecarboxamide
Purity:
≥98%
Inosine monophosphatase dehydrogenase (IMPDH) inhibitor
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