4 results for "CCK2 Receptor Antagonists Small Molecules and Peptides" in Products
CCK2 Receptor Antagonists: Small Molecules and Peptides
The cholecystokinin2 receptor (CCK2 receptor, CCK-B receptor) is a member of the cholecystokinin receptor group of G-protein-coupled receptors that also includes CCK1. They are located primarily in the brain, spinal cord and stomach where they play a role in anxiety, nociception, neuroleptic activity, gastric acid release, gastric mucosal cell growth and histamine release. The human CCK2 receptor gene has been localized to chromosome 11 (11p15.4).
Highly potent, selective non-peptide CCK2 antagonist
| Chemical Name: | (R)-N-[2,3-Dihydro-1-[2-(2-methylphenyl)-2-oxoethyl]-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl]-N'-(3-methylphenyl)-urea |
| Purity: | ≥98% (HPLC) |
Selective CCK2 antagonist
| Chemical Name: | N-[(3R)-2,3-Dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl]-N'-(3-methylphenyl)urea |
| Purity: | ≥98% (HPLC) |
Selective CCK2 antagonist
| Chemical Name: | (4S,5R)-N-(4-Bromophenyl)-3-oxo-4,5-diphenyl-1-pyrazolidinecarboxamide |
| Purity: | ≥98% (HPLC) |
Potent and selective CCK2 antagonist
| Alternate Names: | PD 134308 |
| Chemical Name: | 4-[[(1R)-2-[[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-2-[[(tricyclo[3.3.1.13,7]dec-2-yloxy)carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoic acid |
| Purity: | ≥98% (HPLC) |
