Cannabinoid R1/CB1 Receptor Ligand: Small Molecules and Peptides
Cannabinoid Receptors are seven-pass transmembrane proteins that belong to the rhodopsin family of G protein-coupled receptors. There are at least two types of Cannabinoid receptors, CB1R and CB2R, which are activated by a family of endogenous arachidonic acid derivatives, such as the endocannabinoids and D9-THC. CB1R is expressed in the central nervous system and upper GI tract, while CB2R is expressed by selected neuronal cell types and hematopoietic cells.
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Cannabinoid R1/CB1 Receptor Ligand: Small Molecules and Peptides
Cannabinoid Receptors are seven-pass transmembrane proteins that belong to the rhodopsin family of G protein-coupled receptors. There are at least two types of Cannabinoid receptors, CB1R and CB2R, which are activated by a family of endogenous arachidonic acid derivatives, such as the endocannabinoids and D9-THC. CB1R is expressed in the central nervous system and upper GI tract, while CB2R is expressed by selected neuronal cell types and hematopoietic cells.
Potent and selective CB2 partial agonist; orally biovailable
| Chemical Name: | 3-Cyclopropyl-1-[[4-[6-[(1,1-dioxido-4-thiomorpholinyl)methyl]-5-fluoro-2-pyridinyl]phenyl]methyl]-2,4-imidazolidinedione hydrochloride |
| Purity: | ≥98% (HPLC) |
