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6 results for "aurora-kinase-inhibitors&view=expanded" in Products

Inhibits Aurora kinase B

Chemical Name:
N-[4-[[6-Methoxy-7-[3-(4-morpholinyl)propoxy]-4-quinazolinyl]amino]phenyl]benzamide
Purity:
≥98%
Inhibits Aurora kinase B

Potent pan-Aurora kinase inhibitor

Chemical Name:
N-[4-[[3-(2-Amino-4-pyrimidinyl)-2-pyridinyl]oxy]phenyl]-4-(4-methyl-2-thienyl)-1-phthalazinamine
Purity:
≥98%
Potent and selective pan-Aurora kinases inhibitor

Potent, selective Aurora kinase A inhibitor

Chemical Name:
2-[(5-Hydroxy-1,5-dimethylhexyl)amino]-4-methyl-6-[(5-methyl-1H-pyrazol-3-yl)amino]-3-pyridinecarbonitrile hydrochloride
Purity:
≥98%
Potent, selective Aurora kinase A inhibitor

Potent Aurora kinase B inhibitor

Chemical Name:
N-[2,3-Dihydro-2-oxo-3-[(3Z)-phenyl[[4-(1-piperidinylmethyl)phenyl]amino]methylene]-1H-indol-5-yl]-ethanesulfonamide hydrochloride
Purity:
≥98%
Potent Aurora kinase B inhibitor

JAK2, FLT3 and TrkA inhibitor; also inhibits AurA and AurB

Alternate Names:
CEP-701
Chemical Name:
(9S,10S,12R)-2,3,9,10,11,12-Hexahydro-10-hydroxy-10-(hydroxymethyl)-9-methyl-9,12-epoxy-1H-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocin-1-one
Purity:
≥98%
JAK2, FLT3 and TrkA inhibitor; also inhibits AurA and AurB

PDPK1 (PDK1) inhibitor

Chemical Name:
N-[3-[[5-Iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide
Purity:
≥98%
PDPK1 (PDK1) inhibitor
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