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5 results for "additional-p53-related-compounds&view=expanded" in Products

Restores mutant p53 activity; proapoptotic

Chemical Name:
1-[(1-Oxopropoxy)methyl]-1H-pyrrole-2,5-dione
Restores mutant p53 activity; proapoptotic

Restores mutant p53 activity

Alternate Names:
APR-246
Chemical Name:
2-(Hydroxymethyl)-2-(methoxymethyl)-1-azabicyclo[2.2.2]octan-3-one
Purity:
≥98%
Restores mutant p53 activity

p53 inhibitor. Also aryl hydrocarbon receptor agonist

Chemical Name:
1-(4-Methylphenyl)-2-(4,5,6,7-tetrahydro-2-imino-3(2H)-benzothiazolyl)ethanone hydrobromide
p53 inhibitor. Also aryl hydrocarbon receptor agonist

Selective exportin-1 (XPO1/CRM1) inhibitor

Chemical Name:
(2Z)-3-[3-[3,5-Bis(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl]-2-propenoic acid 2-(2-pyridinyl)hydrazide
Purity:
≥98%
Selective exportin-1 (XPO1/CRM1) inhibitor

RNA polymerase I inhibitor; also p53 pathway activator

Chemical Name:
N-[2-(Dimethylamino)ethyl]-12-oxo-12H-benzo[g]pyrido[2,1-b]quinazoline-4-carboxamide
Purity:
≥98%
RNA polymerase I inhibitor; also p53 pathway activator
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