Proxyfan oxalate

Tocris Bioscience, part of Bio-Techne | Catalog # 2477

High affinity H3 ligand
Discontinued Product
2477 has been discontinued. View all Histamine H3 Receptor Agonists products.

Key Product Details

Description

High affinity H3 ligand

View all Histamine H3 Receptor Agonists »

Product Description

Proxyfan oxalate is a high affinity histamine H3 receptor ligand (pKi = 8.62) that acts as a protean agonist at recombinant and native receptors. In functional studies, activity ranges from full agonist to inverse agonist depending on system used. Displays partial agonist effects on cAMP inhibition and MAPK activity, neutral antagonist activity on histamine release and partial inverse agonism of [3H]-arachidonic acid release.

Product Specifications

Molecular Weight

306.32

Formula

C13H16N2O.C2H2O4

Storage

Desiccate at RT

Purity

≥98% (HPLC)

Chemical Name

4-[3-(Phenylmethoxy)propyl]-1H-imidazole oxalate

CAS Number

1620017-81-3

PubChem ID

76900838

InChI Key

QVMZCQMJBQSPSW-UHFFFAOYSA-N

SMILES

OC(=O)C(O)=O.C(COCC1=CC=CC=C1)CC1=CN=CN1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 33.23 100
DMSO 33.24 100

Preparing Stock Solutions for Proxyfan oxalate

The following data is based on the product molecular weight 306.32

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 3.26 mL 16.32 mL 32.65 mL
5 mM 0.65 mL 3.26 mL 6.53 mL
10 mM 0.33 mL 1.63 mL 3.26 mL
50 mM 0.07 mL 0.33 mL 0.65 mL

Calculators

Molarity Calculator

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Reconstitution Calculator

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Background References

References are publications that support the biological activity of the product.

Product Documents for Proxyfan oxalate

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Proxyfan oxalate

For research use only

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