Immethridine dihydrobromide

Name: Immethridine dihydrobromide
Brand: Tocris Bioscience
SKU: 2315
Rating: 5 (1 reviews)

Tocris Bioscience, part of Bio-Techne | Catalog # 2315

(1)

Citations (7)

COA / SDS

Potent H3 agonist, highly selective over H4

Discontinued Product

2315 has been discontinued. View all Histamine H3 Receptor Agonists products.

Key Product Details

Description:	Potent H₃ agonist, highly selective over H₄
Chemical Name:	4-(1H-Imidazol-4-ylmethyl)pyridine dihydrobromide
Purity:	≥99% (HPLC)
Molecular Weight:	321.01

View Full Technical Details for Immethridine dihydrobromide

Technical Data
Citations / Reviews (1)

Biological Activity for Immethridine dihydrobromide

Immethridine dihydrobromide is a potent and highly selective histamine H₃ receptor agonist (pEC₅₀ = 9.74) that displays 300-fold selectivity over the H₄ receptor (pK_i values are 9.07 and 6.61 respectively). Does not bind to H₁ or H₂ receptors at concentrations up to 10 μM..

Technical Data for Immethridine dihydrobromide

M. Wt	321.01
Formula	C₉H₉N₃.2HBr
Storage	Desiccate at RT
Purity	≥99% (HPLC)
CAS Number	699020-93-4
PubChem ID	16759172
InChi Key	CYNKWHIKNDIVDR-UHFFFAOYSA-N
Smiles	Br.Br.C(C1=CN=CN1)C1=CC=NC=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

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References for Immethridine dihydrobromide

References are publications that support the biological activity of the product.

Kitbunnadaj Identification of 4-(1H-imidazol-4(5)-ylmethyl)pyridine (immethridine) as a novel, potent, and highly selective histamine H₃ receptor agonist. J.Med.Chem. 2004 PMID: 15115383

Immethridine dihydrobromide

Tocris Bioscience, part of Bio-Techne | Catalog # 2315

Key Product Details

Biological Activity for Immethridine dihydrobromide

Technical Data for Immethridine dihydrobromide

Molarity Calculator

Dilution Calculator

Reconstitution Calculator

References for Immethridine dihydrobromide

Product Documents for Immethridine dihydrobromide

COA

Certificate of Analysis

SDS

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