TM 5275 sodium salt
Tocris Bioscience, part of Bio-Techne | Catalog # 5769
Plasminogen activator inhibitor-1 (PAI-1) inhibitor; orally bioavailable
Key Product Details
Description
Plasminogen activator inhibitor-1 (PAI-1) inhibitor; orally bioavailable
Product Description
TM 5275 sodium salt is a plasminogen activator inhibitor-1 (PAI-1) inhibitor. Orally bioavailable.Product Specifications
Molecular Weight
543.97
Formula
C28H27ClN3NaO5
Storage
Store at +4°C
Purity
≥98% (HPLC)
Chemical Name
5-Chloro-2-[[2-[2-[4-(Diphenylmethyl)-1-piperazinyl]-2-oxoethoxy]acetyl]amino]benzoic acid sodium salt
CAS Number
1103926-82-4
PubChem ID
53240409
InChI Key
JSHSGBIWNPQCQZ-UHFFFAOYSA-M
SMILES
O=C(COCC(NC4=C(C(O[Na])=O)C=C(Cl)C=C4)=O)N1CCN(C(C3=CC=CC=C3)C2=CC=CC=C2)CC1
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Solubility
| Solvent | Max Conc. mg/mL | Max Conc. mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 54.4 | 100 |
Preparing Stock Solutions
for TM 5275 sodium salt
The following data is based on the product molecular weight 543.97
Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.84 mL | 9.19 mL | 18.38 mL |
| 5 mM | 0.37 mL | 1.84 mL | 3.68 mL |
| 10 mM | 0.18 mL | 0.92 mL | 1.84 mL |
| 50 mM | 0.04 mL | 0.18 mL | 0.37 mL |
Calculators
Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Background References
References are publications that support the biological activity of the product.
- Yamaoka Structure-activity relationships of new N-acylanthranilic acid derivatives as plasminogen activator inhibitor-1 inhibitors. Chem.Pharm.Bull. 2011 PMID: 21297302
Product Specific Notices for TM 5275 sodium salt
For research use only
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