TCS 2510
Tocris Bioscience, part of Bio-Techne | Catalog # 4069
Selective EP4 agonist
Product Description
TCS 2510 is a highly selective EP4 agonist (EC50 = 2.5 nM; Ki = 1.2 nM). Displays no significant binding at other prostaglandin receptors at concentrations up to 14 μM.Product Specifications
Molecular Weight
383.49
Formula
C21H29N5O2
Storage
Store at -20°C
Purity
≥98% (HPLC)
Chemical Name
(5R)-5-[(3S)-3-Hydroxy-4-phenyl-1-buten-1-yl]-1-[6-(2H-tetrazol-5-yl)hexyl]-2-pyrrolidinone
CAS Number
346673-06-1
PubChem ID
9864831
InChI Key
JWYPJSNXPZTEHL-VJKINUSGSA-N
SMILES
O=C1N(CCCCCCC2=NN=NN2)[C@@H](/C=C/[C@H](CC3=CC=CC=C3)O)CC1
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Solubility
| Solubility | Soluble in ethanol (supplied pre-dissolved in anhydrous ethanol, 5mg/ml) |
Calculators
Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Background References
References are publications that support the biological activity of the product.
- Billot Discovery of a potent and selective agonist of the prostaglandin EP4 receptor. Bioorg.Med.Chem.Lett.
Product Specific Notices for TCS 2510
For research use only
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