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SB 699551

Tocris Bioscience, part of Bio-Techne | Catalog # 3188

Selective 5-ht5a antagonist
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3188/50
3188/10

Key Product Details

Description

Selective 5-ht5a antagonist

Product Description

SB 699551 is a selective 5-ht5a receptor antagonist (pKi values are 8.3, < 6.0, < 6.0, < 6.0, < 5.5 and < 5.5 for 5-ht5a, 5-HT1B/D, 5-HT2A, 5-HT2C, 5-HT1A and 5-HT7 receptors respectively).

Licensing Information

Sold for research purposes under agreement from GlaxoSmithKline

Product Specifications

Molecular Weight

584.66

Formula

C34H45N3O.2HCl

Storage

Store at +4°C

Purity

≥98% (HPLC)

Chemical Name

N-[2-(Dimethylamino)ethyl]-N-[[4'-[[(2-phenylethyl)amino]methyl][1,1'-biphenyl]-4-yl]methyl]cyclopentanepropanamide dihydrochloride

CAS Number

864741-95-7

PubChem ID

11983346

InChI Key

QJMKBIHLMPTYTI-UHFFFAOYSA-N

SMILES

O=C(CCC4CCCC4)N(CCN(C)C)CC(C=C2)=CC=C2C1=CC=C(CNCCC3=CC=CC=C3)C=C1.Cl.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 14.62 25
Ethanol 5.85 10

Preparing Stock Solutions for SB 699551

The following data is based on the product molecular weight 584.66

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.25 mM 6.84 mL 34.21 mL 68.42 mL
1.25 mM 1.37 mL 6.84 mL 13.68 mL
2.5 mM 0.68 mL 3.42 mL 6.84 mL
12.5 mM 0.14 mL 0.68 mL 1.37 mL

Calculators

Molarity Calculator

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Dilution Calculator

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Reconstitution Calculator

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Background References

References are publications that support the biological activity of the product.

Product Documents for SB 699551

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for SB 699551

For research use only

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