SB 216641 hydrochloride

Tocris Bioscience, part of Bio-Techne | Catalog # 1242

Selective h5-HT1B antagonist
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Key Product Details

Description

Selective h5-HT1B antagonist

View all 5-HT1B Receptor Antagonists »

Product Description

SB 216641 hydrochloride is a selective h5-HT1B antagonist with approximately 25-fold selectivity over h5-HT1D and little or no affinity for a range of other receptor types.

Licensing Information

Sold with the permission of GlaxoSmithKline

Product Specifications

Molecular Weight

523.03

Formula

C28H30N4O4.HCl

Storage

Store at RT

Purity

≥98% (HPLC)

Chemical Name

N-[3-[3-(Dimethylamino)ethoxy]-4-methoxyphenyl]-2'-methyl-4'-(5-methyl-1,2,4-oxadiazol-3-yl)-[1,1'-biphenyl]-4-carboxamide hydrochloride

CAS Number

193611-67-5

PubChem ID

10392025

InChI Key

JPBMDMNORXKGHZ-UHFFFAOYSA-N

SMILES

Cl.COC1=C(OCCN(C)C)C=C(NC(=O)C2=CC=C(C=C2)C2=CC=C(C=C2C)C2=NOC(C)=N2)C=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 26.15 50

Preparing Stock Solutions for SB 216641 hydrochloride

The following data is based on the product molecular weight 523.03

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.5 mM 3.82 mL 19.12 mL 38.24 mL
2.5 mM 0.76 mL 3.82 mL 7.65 mL
5 mM 0.38 mL 1.91 mL 3.82 mL
25 mM 0.08 mL 0.38 mL 0.76 mL

Calculators

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Reconstitution Calculator

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Background References

References are publications that support the biological activity of the product.

Product Documents for SB 216641 hydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for SB 216641 hydrochloride

For research use only

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