Sarpogrelate hydrochloride

Tocris Bioscience, part of Bio-Techne | Catalog # 3739

Selective 5-HT2A antagonist
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Key Product Details

Description

Selective 5-HT2A antagonist

Alternative Names

MCI 9042

View all 5-HT2A Receptor Antagonists »

Product Description

Sarpogrelate hydrochloride is a selective 5-HT2A receptor antagonist (pKi values are 8.52, 7.43 and 6.57 for 5-HT2A, 5-HT2C and 5-HT2B receptors respectively). Displays selectivity over 5-HT1, 5-HT3, 5-HT4 H1, H2, M3, α1-adrenergic, α2-adrenergic and β-adrenergic receptors. Displays cardioprotective activity in vivo.

Product Specifications

Molecular Weight

465.97

Formula

C24H31NO6.HCl

Storage

Desiccate at RT

Purity

≥98% (HPLC)

Chemical Name

Succinic acid mono-(1-dimethylaminomethyl-2-(2-[2-(3-methoxyphenyl)ethyl]phenoxy)ethyl) ester hydrochloride

CAS Number

135159-51-2

PubChem ID

444005

InChI Key

POQBIDFFYCYHOB-UHFFFAOYSA-N

SMILES

O=C(CCC(O)=O)OC(CN(C)C)COC1=CC=CC=C1CCC2=CC(OC)=CC=C2.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 11.65 25
DMSO 46.6 100

Preparing Stock Solutions for Sarpogrelate hydrochloride

The following data is based on the product molecular weight 465.97

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.15 mL 10.73 mL 21.46 mL
5 mM 0.43 mL 2.15 mL 4.29 mL
10 mM 0.21 mL 1.07 mL 2.15 mL
50 mM 0.04 mL 0.21 mL 0.43 mL

Calculators

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Product Documents for Sarpogrelate hydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Sarpogrelate hydrochloride

For research use only

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