PDZ1 Domain inhibitor peptide

Tocris Bioscience, part of Bio-Techne | Catalog # 2207

Disrupts interaction between GluK2 and PSD-95 PDZ1 domain
Discontinued Product
2207 has been discontinued. View all Kainate Receptor Peptides products.

Key Product Details

Description

Disrupts interaction between GluK2 and PSD-95 PDZ1 domain

View all Kainate Receptor Peptides »

Product Description

PDZ1 Domain inhibitor peptide is a novel cyclic peptide that disrupts interaction between GluK2 (formerlyy GluR6) and the postsynaptic density protein 95 (PSD-95). Competes with the C-terminus of GluK2 for binding to the PDZ1 domain of PSD-95. Inhibits clustering of kainate receptors.

Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions.

Product Specifications

Molecular Weight

819.95

Formula

C38H61N9O11

Storage

Desiccate at -20°C

CAS Number

1315378-73-4

PubChem ID

90488746

InChI Key

XXRRADBJCXMGOW-RMLJCASOSA-N

SMILES

[H]N[C@@H](CC1=CC=C(O)C=C1)C(=O)N[C@@H](CCCCN)C(=O)N[C@H]1CCCCNC(=O)CC[C@H](NC(=O)[C@@H](NC1=O)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)N[C@@H](C(C)C)C(O)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solubility Soluble to 4mg/ml in DMSO and to 1mg/ml in 5% acetonitrile / water

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Background References

References are publications that support the biological activity of the product.

Product Documents for PDZ1 Domain inhibitor peptide

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for PDZ1 Domain inhibitor peptide

For research use only

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