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Ocinaplon

Tocris Bioscience, part of Bio-Techne | Catalog # 4410

GABAA modulator; anxiolytic
Discontinued Product
4410 has been discontinued. View all GABA-A Receptor Modulators products.

Key Product Details

Description

GABAA modulator; anxiolytic

Product Description

Ocinaplon is a modulator of GABAA receptors. Displays modest selectivity for GABAA α1 receptors; displays partial agonist activity at α2-, α3- and α5-containing receptors. Exhibits anxiolytic activity.

Product Specifications

Molecular Weight

301.30

Formula

C17H11N5O

Storage

Store at +4°C

Purity

≥98% (HPLC)

Chemical Name

2-Pyridinyl[7-(4-pyridinyl)pyrazolo[1,5-a]pyrimidin-3-yl]methanone

CAS Number

96604-21-6

PubChem ID

216456

InChI Key

OQJFBUOFGHPMSR-UHFFFAOYSA-N

SMILES

O=C(C4=CC=CC=N4)C2=C1N=CC=C(C3=CC=NC=C3)N1N=C2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
2eq.HCl 30.13 100
DMSO 3.01 10

Preparing Stock Solutions for Ocinaplon

The following data is based on the product molecular weight 301.30

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 3.32 mL 16.59 mL 33.19 mL
5 mM 0.66 mL 3.32 mL 6.64 mL
10 mM 0.33 mL 1.66 mL 3.32 mL
50 mM 0.07 mL 0.33 mL 0.66 mL

Calculators

Molarity Calculator

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Dilution Calculator

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Reconstitution Calculator

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Background References

References are publications that support the biological activity of the product.

Product Documents for Ocinaplon

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Ocinaplon

For research use only

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