Desmethyl-YM 298198

Name: Desmethyl-YM 298198
Brand: Tocris Bioscience
SKU: 2447

Tocris Bioscience, part of Bio-Techne | Catalog # 2447

COA / SDS

Derivative of mGlu1 antagonist YM 298198 (Cat. No. 2448)

Discontinued Product

2447 has been discontinued. View all Group I mGluR Antagonists products.

Key Product Details

Description:	Derivative of mGlu₁antagonist YM 298198 (Cat. No. 2448)
Chemical Name:	6-Amino-N-cyclohexyl-3-methylthiazolo[3,2-a]benzimidazole-2-carboxamide hydrochloride
Purity:	≥98% (HPLC)
Molecular Weight:	364.89

View Full Technical Details for Desmethyl-YM 298198

Technical Data
Citations

Biological Activity for Desmethyl-YM 298198

Desmethyl-YM 298198 is a derivative of the mGlu₁-selective antagonist YM 298198 (Cat. No. 2448).

Licensing Information

Sold with the permission of Astellas Pharma Inc.

Technical Data for Desmethyl-YM 298198

M. Wt	364.89
Formula	C₁₇H₂₀N₄OS.HCl
Storage	Desiccate at RT
Purity	≥98% (HPLC)
CAS Number	1177767-57-5
PubChem ID	16759180
InChi Key	SWKZWXJQIDXGLX-UHFFFAOYSA-N
Smiles	Cl.CC1=C(SC2=NC3=CC=C(N)C=C3N12)C(=O)NC1CCCCC1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

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References for Desmethyl-YM 298198

References are publications that support the biological activity of the product.

Kohara Radioligand binding properties and pharmacological characterization of 6-Amino-N-cyclohexyl-N,3-dimethyl-thiazolo[3,2-a]-benzimidazole-2-carboxamide (YM-298198), a high-affinity, selective and noncompetitive antagonist of metabo J.Pharmacol.Exp.Ther. 2005 PMID: 15976016