CYN 154806
Tocris Bioscience, part of Bio-Techne | Catalog # 1843
Selective sst2 antagonist
Key Product Details
Description
Selective sst2 antagonist
Product Description
CYN 154806 is a potent and selective somatostatin sst2 receptor antagonist. pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively.Product Specifications
Molecular Weight
1197.35
Formula
C56H68N12O14S2
Storage
Store at -20°C
Purity
≥95% (HPLC)
CAS Number
183658-72-2
PubChem ID
16133842
InChI Key
RDTVTSXTFYXNSG-HDNDNHAUSA-N
SMILES
C[C@@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CC2=CNC3=C2C=CC=C3)NC(=O)[C@H](CC2=CC=C(O)C=C2)NC(=O)[C@@H](CSSC[C@H](NC1=O)C(=O)N[C@H](CC1=CC=C(O)C=C1)C(N)=O)NC(=O)[C@H](CC1=CC=C(C=C1)[N+]([O-])=O)NC(C)=O
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Solubility
| Solubility | Soluble to 1mg/ml in water |
Calculators
Molarity Calculator
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Background References
References are publications that support the biological activity of the product.
- Feniuk Selective somatostatin sst2 receptor blockade with the novel cyclic octapeptide, CYN-154806. Neuropharmacology 2000 PMID: 10818260
- Hannon Drug design at peptide receptors. Somatostatin receptor ligands. J.Mol.Neurosci. 2002 PMID: 11931345
- Bass Identification and characterization of novel somatostatin antagonists. Mol.Pharmacol. 1996 PMID: 8863814
Product Specific Notices for CYN 154806
For research use only
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