CGS 12066B dimaleate

Tocris Bioscience, part of Bio-Techne | Catalog # 0638

5-HT1B agonist
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Key Product Details

Description

5-HT1B agonist

View all 5-HT1B Receptor Agonists »

Product Description

CGS 12066B dimaleate is a 5-HT1B full agonist, 10-fold selective over 5-HT1A and 1000-fold selective over 5-HT2C receptors. Centrally active following systemic administration.

Product Specifications

Molecular Weight

566.49

Formula

C17H17F3N4.2C4H4O4

Storage

Store at RT

Purity

≥98% (HPLC)

Chemical Name

7-Trifluoromethyl-4-(4-methyl-1-piperazinyl)pyrrolo[1,2-a]-quinoxaline dimaleate

CAS Number

109028-10-6

PubChem ID

9915956

InChI Key

HTEVMLYDEWVIQE-SPIKMXEPSA-N

SMILES

O=C(O)/C=C\C(O)=O.O=C(O)/C=C\C(O)=O.FC(C1=CC3=C(N2C=CC=C2C(N4CCN(CC4)C)=N3)C=C1)(F)F

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 2.83 5
DMSO 22.66 40

Preparing Stock Solutions for CGS 12066B dimaleate

The following data is based on the product molecular weight 566.49

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.4 mM 4.41 mL 22.07 mL 44.13 mL
2 mM 0.88 mL 4.41 mL 8.83 mL
4 mM 0.44 mL 2.21 mL 4.41 mL
20 mM 0.09 mL 0.44 mL 0.88 mL

Calculators

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Reconstitution Calculator

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Background References

References are publications that support the biological activity of the product.

Product Documents for CGS 12066B dimaleate

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for CGS 12066B dimaleate

For research use only

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