BRL 52537 hydrochloride
Tocris Bioscience, part of Bio-Techne | Catalog # 0699
Potent and selective κ agonist
Discontinued Product
0699 has been discontinued.
View all Kappa Opioid Receptor Agonists products.
Key Product Details
Description
Potent and selective κ agonist
Product Description
The most κ/μ-selective and among the most potent κ ligands known (25 times more potent than morphine in vivo).Licensing Information
Sold with the permission of GlaxoSmithKlineProduct Specifications
Molecular Weight
391.77
Formula
C18H24Cl2N2O.HCl
Storage
Store at RT
Purity
≥98% (HPLC)
Chemical Name
(±)-1-(3,4-Dichlorophenyl)acetyl-2-(1-pyrrolidinyl)methylpiperidine hydrochloride
CAS Number
112282-24-3
PubChem ID
11315337
InChI Key
NGVLSOWJSUUYDE-UHFFFAOYSA-N
SMILES
Cl.ClC1=CC=C(CC(=O)N2CCCCC2CN2CCCC2)C=C1Cl
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Solubility
| Solvent | Max Conc. mg/mL | Max Conc. mM | |
|---|---|---|---|
| Solubility | |||
| water | 1.96 | 5 with gentle warming |
Preparing Stock Solutions
for BRL 52537 hydrochloride
The following data is based on the product molecular weight 391.77
Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.05 mM | 51.05 mL | 255.25 mL | 510.50 mL |
| 0.25 mM | 10.21 mL | 51.05 mL | 102.10 mL |
| 0.5 mM | 5.11 mL | 25.53 mL | 51.05 mL |
| 2.5 mM | 1.02 mL | 5.11 mL | 10.21 mL |
Calculators
Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Background References
References are publications that support the biological activity of the product.
- Vecchietti (2S)-1-(Arylacetyl)-2-(aminomethyl)piperidine derivatives: novel, highly selective κ opioid analgesics. J.Med.Chem. 1991 PMID: 1846921
Product Specific Notices for BRL 52537 hydrochloride
For research use only
Loading...
Loading...