3-Bromocytisine

Tocris Bioscience, part of Bio-Techne | Catalog # 3549

Potent α4β4, α4β2 and α7 nAChR agonist
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Key Product Details

Description

Potent α4β4, α4β2 and α7 nAChR agonist

View all Additional Nicotinic Receptor Agonists »

Product Description

3-Bromocytisine is a potent agonist of α4β4, α4β2 and α7 nACh receptors (IC50 values are 0.28, 0.30 and 31.6 nM respectively). Displays different effects on high (HS) and low (LS) ACh sensitivity α4β2 nAChRs (EC50 values are 0.008 and 0.05 μM respectively).

Product Specifications

Molecular Weight

269.14

Formula

C11H13BrN2O

Storage

Store at -20°C

Purity

≥98% (HPLC)

Chemical Name

(1R,5S)-9-Bromo-1,2,3,4,5,6-hexahydro-1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one

CAS Number

207390-14-5

PubChem ID

15519735

InChI Key

DWDCLEHDNICBMI-JGVFFNPUSA-N

SMILES

O=C2N1C[C@@]([H])(C3)CNC[C@@]([H])3C1=CC=C2Br

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 26.91 100
DMSO 26.91 100

Preparing Stock Solutions for 3-Bromocytisine

The following data is based on the product molecular weight 269.14

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 3.72 mL 18.58 mL 37.16 mL
5 mM 0.74 mL 3.72 mL 7.43 mL
10 mM 0.37 mL 1.86 mL 3.72 mL
50 mM 0.07 mL 0.37 mL 0.74 mL

Calculators

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Reconstitution Calculator

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Background References

References are publications that support the biological activity of the product.

Product Documents for 3-Bromocytisine

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for 3-Bromocytisine

For research use only

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