CELT-211

CELT-211 is a potent and selective fluorescent h5HT_2B serotonin receptor ligand. It shows full selectivity for h5HT_2B over h5HT_2A, h5HT_2C (K_i values is 56.3 nM for h5HT_2B receptors in radioligand binding assay). Excitation and emission maxima (λ) are 589 and 616 nm, respectively. Wavelengths are compatible with use as an acceptor dye in TR-FRET assays, together with the CoraFluor™ 1 (Cat. No. 7920) TR-FRET donor.

Add 82 μL of assay buffer containing 1% of DMSO to obtain a 100 μM stock solution, and use 250 nM as a working concentration.

Sold under license from Celtarys Research