Skip to main content

21 results for "Integrin Receptor Inhibitors" in Products

Integrin Receptor Inhibitors

Glycoprotein IIb/IIIa (integrin αIIbβ3) receptor antagonist. Antithrombotic

Chemical Name:
4-[4-[4-(Aminoiminomethyl)phenyl]-1-piperazinyl]-1-piperidineacetic acid trihydrochloride
Purity:
≥98%
Glycoprotein IIb/IIIa (integrin αIIbβ3) receptor antagonist. Antithrombotic

Selective α4β1 (VLA-4) inhibitor

Purity:
≥95%
Selective α4β1 (VLA-4) inhibitor

Selective inhibitor of integrin α2β1

Chemical Name:
1-(4-Fluorophenyl)-N-methyl-N-[4[[(phenylamino)carbonyl]amino]phenyl]-1H-pyrazole-4-sulfonamide
Purity:
≥98%
Selective inhibitor of integrin α2β1

Integrin binding sequence; inhibits integrin receptor function

Purity:
≥95%
Integrin binding sequence; inhibits integrin receptor function

Dual α9β1/α4β1 integrin inhibitor; preferentially mobilizes HSCs

Chemical Name:
N-(Benzenesulfonyl)-L-prolyl-L-O-(1-pyrrolidinylcarbonyl)tyrosine sodium salt
Purity:
≥98%
Dual α9β1/α4β1 integrin inhibitor; preferentially mobilizes HSCs

Highly potent and selective inhibitor of integrin α4β1 (VLA-4)

Chemical Name:
(2S)-2-[[[(2S)-1-[(3,5-Dichlorophenyl)sulfonyl]-2-pyrrolidinyl]carbonyl]amino]-4-[[(2S)-4-methyl-2-[methyl[2-[4-[[[(2-methylphenyl)amino]carbonyl]amino]phenyl]acetyl]amino]-1-oxopentyl]amino]butanoic acid
Purity:
≥98%
Highly potent and selective inhibitor of integrin α4β1 (VLA-4)

Potent α2β1 inhibitor; displays antithrombotic activity in vivo

Chemical Name:
N-[[(4R)-5,5-Dimethyl-3-(phenylsulfonyl)-4-thiazolidinyl]carbonyl]-3-[[[(phenylmethyl)amino]carbonyl]amino]-L-alanine
Purity:
≥98%
Potent α2β1 inhibitor; displays antithrombotic activity in vivo

Potent and selective α1β1 inhibitor

Purity:
≥95%
Potent and selective α1β1 inhibitor

Potent negative allosteric modulator of LFA-1

Chemical Name:
(5R)-5-[(4-Bromophenyl)methyl]-3-(3,5-dichlorophenyl)-1,5-dimethyl-2,4-imidazolidinedione
Purity:
≥98%
Potent negative allosteric modulator of LFA-1

Potent and selective inhibitor of integrins αvβ3 and αvβ5

Alternate Names:
EMD121974
Purity:
≥95%
Potent and selective inhibitor of integrins αvβ3 and αvβ5

α5β1 integrin receptor antagonist

Purity:
≥95%
α5β1 integrin receptor antagonist

αVβ3 and glycoprotein IIb/IIIa (integrin αIIbβ3) inhibitor

Purity:
≥95%
αVβ3 and glycoprotein IIb/IIIa (integrin αIIbβ3) inhibitor

α4β1 (VLA-4) antagonist

Chemical Name:
1-[[(3S)-4-[2-[4-[[[(2-Methylphenyl)amino]carbonyl]amino]phenyl]acety]l-3-morpholinyl]carbonyl]-4-piperidinediacetic acid
Purity:
≥98%
α4β1 (VLA-4) antagonist

Potent inhibitor of the LFA-1/ICAM-1 interaction

Chemical Name:
(2E)-1-(4-Acetyl-1-piperazinyl)-3-[4-[[2-(1-methylethyl)phenyl]thio]-3-nitrophenyl]-2-propen-1-one
Purity:
≥98%
Potent inhibitor of the LFA-1/ICAM-1 interaction

Potent inhibitor of the LFA-1/ICAM interaction

Chemical Name:
6-[(5S,9R)-9-(4-Cyanophenyl)-3-(3,5-dichlorophenyl)-1-methyl-2,4-dioxo-1,3,7-triazaspiro[4,4]non-7-yl]-3-pyridinecarboxylic acid
Purity:
≥98%
Potent inhibitor of the LFA-1/ICAM interaction

Potent and selective α5β1 integrin inhibitor

Chemical Name:
N-(2,6-Dimethylbenzoyl)-O-[3-(2-pyridinylamino)propyl]-L-tyrosine
Purity:
≥98%
Potent and selective α5β1 integrin inhibitor

α2 integrin inhibitor; anti-angiogenic

Chemical Name:
3-Cyano-N-(3-cyano-4-methyl-1H-indol-7-yl)benzenesulfonamide
Purity:
≥98%
α2 integrin inhibitor; anti-angiogenic

Potent integrin α4β7 and α4β1 (VLA-4) antagonist; orally bioavailable

Chemical Name:
(αS)-α-[(2,6-Dichlorobenzoyl)amino]-2',6'-dimethoxy[1,1'-biphenyl]-4-propanoic acid
Purity:
≥98%
Potent integrin α4β7 and α4β1 (VLA-4) antagonist; orally bioavailable

Potent αv integrin inhibitor

Chemical Name:
3-[[2,5-Dimethyl-6-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)-1-piperidinyl]-4-pyrimidinyl]amino]-N-[(4-methoxyphenyl)sulfonyl]-L-alanine
Purity:
≥97%
Potent αv integrin inhibitor

ανβ6 integrin inhibitor

Chemical Name:
N-[1-Oxo-5-(2-pyridinylamino)pentyl]-O-(phenylmethyl)-L-seryl-3-(3,5-dichlorophenyl)-β-alanine hydrochloride
Purity:
≥98%
ανβ6 integrin inhibitor

Minimal recognition sequence for integrin binding; potent integrin inhibitor

Purity:
≥95%
Minimal recognition sequence for integrin binding; potent integrin inhibitor
Results Per Page
5 10 25 50
  • / 1