Kainate Receptor Antagonists: Small Molecules and Peptides
13 results for "Kainate Receptor Antagonists Small Molecules and Peptides" in Products
13 results for "Kainate Receptor Antagonists Small Molecules and Peptides" in Products
Kainate Receptor Antagonists: Small Molecules and Peptides
Potent and selective non-NMDA iGluR antagonist
| Alternate Names: | Cyanquixaline |
| Chemical Name: | 6-Cyano-7-nitroquinoxaline-2,3-dione |
| Purity: | ≥98% (HPLC) |
Potent non-NMDA iGluR antagonist; more water soluble form of CNQX (Cat. No. 0190)
| Chemical Name: | 6-Cyano-7-nitroquinoxaline-2,3-dione disodium |
| Purity: | ≥98% (HPLC) |
Selective non-NMDA iGluR antagonist
| Chemical Name: | 6,7-Dinitroquinoxaline-2,3-dione |
| Purity: | ≥98% (HPLC) |
Potent kainate antagonist; displays selectivity for GluK1-containing receptors
| Chemical Name: | (S)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxy-5-phenylthiophene-3-yl-methyl)-5-methylpyrimidine-2,4-dione |
| Purity: | ≥98% (HPLC) |
Potent and selective kainate antagonist; selective for GluK1-containing receptors
| Chemical Name: | (RS)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxybenzyl)pyrimidine-2,4-dione |
| Purity: | ≥98% (HPLC) |
Non-competitive non-NMDA iGluR antagonist
| Alternate Names: | GYKI 53773,LY 300164 |
| Chemical Name: | (8R)-7-Acetyl-5-(4-aminophenyl)-8,9-dihydro-8-methyl-7H-1,3-dioxolo[4,5-h][2,3]benzodiazepine |
| Purity: | ≥98% (HPLC) |
Selective non-NMDA iGluR antagonist; water-soluble salt of DNQX (Cat. No. 0189)
| Chemical Name: | 6,7-Dinitroquinoxaline-2,3-dione disodium salt |
| Purity: | ≥98% (HPLC) |
GluK1-selective kainate antagonist
| Chemical Name: | (S)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxy-thiophene-3-yl-methyl)-5-methylpyrimidine-2,4-dione |
| Purity: | ≥98% (HPLC) |
GluK1 antagonist; inhibits carbonic anhydrase (CA) II and IV; also positive allosteric modulator of GABAA receptors
| Alternate Names: | Topamax |
| Chemical Name: | 2,3:4,5-Bis-O-(1-methylethylidene)-β-D-fructopyranose sulfamate |
| Purity: | ≥98% (HPLC) |
Non-competitive non-NMDA iGluR antagonist
| Chemical Name: | 1-(4-Aminophenyl)-3-methylcarbamyl-4-methyl-3,4-dihydro-7,8-methylenedioxy-5H-2,3-benzodiazepine hydrochloride |
| Purity: | ≥98% (HPLC) |
Potent and selective kainate antagonist; active enantiomer of UBP 296 (Cat. No. 2078)
| Chemical Name: | (S)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxybenzyl)pyrimidine-2,4-dione |
| Purity: | ≥98% (HPLC) |
Competitive non-NMDA iGluR antagonist
| Alternate Names: | MPQX |
| Chemical Name: | [[3,4-Dihydro-7-(4-morpholinyl)-2,3-dioxo-6-(trifluoromethyl)-1(2H)-quinoxalinyl]methyl]phosphonic acid |
| Purity: | ≥98% (HPLC) |
Dye for assessing cell viability and blood brain barrier permeability; also EAAT inhibitor and iGluR antagonist
| Chemical Name: | 6,6-[(3,3'-Dimethyl[1,1'-biphenyl]-4,4'-diyl)bis(azo)bis[4-amino- 5-hydroxy-1,3-naphthalenedisulphonic acid] tetrasodium salt |
| Purity: | ≥90% (HPLC) |