11 results for "ER beta/NR3A2 Small Molecules and Peptides" in Products
ER beta/NR3A2: Small Molecules and Peptides
Estrogen Receptor beta (ERβ,NR3A2) is a member of the steroid receptor family. The natural ligand for ER is the classical estrogenic compound 17β-estradiol. ERβ is expressed in the granulosa cell layer of primary, secondary and mature follicles in the ovary, in bone, bladder, uterus, testis, epididymis, gastrointestinal tract, kidney, breast, heart, vessel wall, immune system, lung, pituitary, hippocampus and hypothalamus. Roles for ERβ in the reproductive and cardiovascular ...
Highly potent ERβ agonist
| Alternate Names: | Diarylpropionitrile |
| Chemical Name: | 2,3-bis(4-Hydroxyphenyl)-propionitrile |
| Purity: | ≥98% (HPLC) |
Selective ERβ antagonist
| Chemical Name: | 4-[2-Phenyl-5,7-bis(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]phenol |
| Purity: | ≥98% (HPLC) |
Estrogen receptor antagonist
| Alternate Names: | Fulvestrant |
| Chemical Name: | 7α,17β-[9-[(4,4,5,5,5-Pentafluoropentyl)sulfinyl]nonyl]estra-1,3,5(10)-triene-3,17-diol |
| Purity: | ≥98% (HPLC) |
Potent subtype-selective ligand; ERα agonist/ERβ antagonist
| Chemical Name: | (R,R)-5,11-Diethyl-5,6,11,12-tetrahydro-2,8-chrysenediol |
| Purity: | ≥98% (HPLC) |
Estrogen receptor partial agonist/antagonist
| Chemical Name: | 2-[4-[(1Z)-1,2-Diphenyl-1-buten-1-yl]phenoxy]-N,N-dimethylethanamine |
| Purity: | ≥98% (HPLC) |
Metabolite of tamoxifen (Cat. No. 0999)
| Alternate Names: | 4-OH-TAM |
| Chemical Name: | 4-[(1Z)-1-[4-[2-(Dimethylamino)ethoxy]phenyl]-2-phenyl-1-buten-1-yl]phenol |
| Purity: | ≥98% (HPLC) |
Potent ERβ agonist
| Chemical Name: | 7-Ethenyl-2-(3-fluoro-4-hydroxyphenyl)-5-benzoxazolol |
| Purity: | ≥98% (HPLC) |
Estrogen receptor partial agonist/antagonist
| Chemical Name: | (Z)-2-[4-(1,2-Diphenyl-1-butenyl)phenoxy]-N,N-dimethylethanamine citrate |
| Purity: | ≥98% (HPLC) |
Selective estrogen receptor modulator (SERM)
| Alternate Names: | LY 139481,Keoxifene |
| Chemical Name: | [6-Hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]phenyl]-methanone hydrochloride |
| Purity: | ≥98% (HPLC) |
Potent and selective ERβ agonist; neuroprotective
| Chemical Name: | 4-[4,4-Difluoro-1-(2-fluorophenyl)cyclohexyl]phenol |
| Purity: | ≥98% (HPLC) |
EGFR kinase inhibitor. Also estrogen and PPARγ ligand
| Chemical Name: | 5,7-Dihydroxy-3-(4-hydroxyphenyl)-4H-1-benzopyran-4-one |
| Purity: | ≥98% (HPLC) |