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DREADD Activators: Small Molecules and Peptides

11 results for "DREADD Activators Small Molecules and Peptides" in Products

11 results for "DREADD Activators Small Molecules and Peptides" in Products

DREADD Activators: Small Molecules and Peptides

Potent hM3Dq and hM4Di DREADD agonist; water soluble version of DREADD agonist 21 (Cat. No. 5548)

Alternate Names: Compound 21 (water-soluble)
Chemical Name: 11-(1-Piperazinyl)-5H-dibenzo[b,e][1,4]diazepine dihydrochloride
Purity: ≥98% (HPLC)
Potent hM3Dq and hM4Di DREADD agonist; water soluble version of DREADD agonist 21 (Cat. No. 5548)

Potent hM3Dq and hM4Di DREADD agonist; blood brain barrier penetrant

Alternate Names: Compound 21,C21
Chemical Name: 11-(1-Piperazinyl)-5H-dibenzo[b,e][1,4]diazepine
Purity: ≥98% (HPLC)
Potent hM3Dq and hM4Di DREADD agonist; blood brain barrier penetrant

Activator of hM3Dq and hM4Di DREADDs; water soluble version of Clozapine N-oxide (Cat. No. 4936)

Alternate Names: CNO (water-soluble)
Chemical Name: 8-Chloro-11-(4-methyl-4-oxido-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine dihydrochloride
Purity: ≥99% (HPLC)
Activator of hM3Dq and hM4Di DREADDs; water soluble version of Clozapine N-oxide (Cat. No. 4936)

Activator of hM3Dq and hM4Di DREADDs

Alternate Names: CNO
Chemical Name: 8-Chloro-11-(4-methyl-4-oxido-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine
Purity: ≥98% (HPLC)
Activator of hM3Dq and hM4Di DREADDs

High affinity and highly potent activator of hM3Dq and hM4Di DREADDs; rapid blood-brain barrier penetrant

Alternate Names: DCZ
Chemical Name: 11-(4-Methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine
Purity: ≥98% (HPLC)
High affinity and highly potent activator of hM3Dq and hM4Di DREADDs; rapidly blood brain barrier penetrant

High affinity and highly potent hM3Dq and hM4Di DREADD agonist; blood brain barrier penetrant

Chemical Name: 8-Chloro-11-(4-ethylpiperazin-1-yl)-4-fluoro-5H-dibenzo[b,e][1,4]diazepine
Purity: ≥98% (HPLC)
High affinity and highly potent hM3Dq and hM4Di DREADD agonist; blood brain barrier penetrant

Activator of κ-opioid DREADD (KORD)

Chemical Name: (2S,4aR,6aR,7R,9S,10aS,10bR)-2-(3-Furanyl)dodecahydro-9-hydroxy-6a,10b-dimethyl-4,10-dioxo-2H-naphtho[2,1-c]pyran-7-carboxylic acid methyl ester
Purity: ≥98% (HPLC)
Activator of κ-opioid DREADD (KORD)

High affinity and highly potent hM3Dq and hM4Di DREADD agonist; blood brain barrier penetrant

Chemical Name: 8-Chloro-11-(4-ethylpiperazin-1-yl)-1-fluoro-5H-dibenzo[b,e][1,4]diazepine
Purity: ≥98% (HPLC)
High affinity and highly potent hM3Dq and hM4Di DREADD agonist; blood brain barrier penetrant

Potent hM3Dq and hM4Di DREADD agonist in vitro

Chemical Name: 6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine
Purity: ≥99% (HPLC)
Potent hM3Dq and hM4Di DREADD agonist in vitro

Selective orthostatic agonist of hFFA2-DREADDs

Chemical Name: 4-Methoxy-3-methylbenzoic acid
Purity: ≥98% (HPLC)
Selective orthostatic agonist of hFFA2-DREADDs

5-HT2A antagonist; also D2 antagonist; atypical antipsychotic

Chemical Name: 2-Methyl-4-(4-methyl-1-piperazinyl)-10H-thieno[2,3-b][1,5]benzodiazepine
Purity: ≥98% (HPLC)
5-HT2A antagonist; also D2 antagonist; atypical antipsychotic
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