145 results for "Vanilloid R1/TRPV1" in Products
Vanilloid R1/TRPV1 Products
Vanilloid Receptor 1 (VR1) also known as TRPV1 (Transient Receptor Potential Vanilloid 1) and capsaicin receptor, is a 115 kDa integral membrane ion channel that has six transmembrane domains and contains intracellular N-and C-termini. Vanilloid Receptor 1 contributes to normal pain and temperature sensation and also has a sensory-effector function. By alternative splicing, at least three VR1 isoforms are known. The sequence of residues 4 - 21 of rat VR1 is 78% and 28% identical to that of mouse and human VR1, respectively.
Potent TRPV agonist
TRPV agonist
TRPV antagonist; also activator of ENaCδ
Endogenous and non-selective CB agonist
Potent and selective TRPV1 competitive antagonist
Potent and selective TRPV1 antagonist
Chloride channel blocker; TRPV1 modulator; RAD51 recombinase inhibitor
Potent and selective TRPV1 competitive antagonist
Reversible, competitive and potent TRPV1 antagonist
Potent and selective endogenous TRPV1 agonist
TRPV1 antagonist
Potent and selective TRPV1 antagonist
Potent TRPV1 antagonist
Potent TRPV1 antagonist