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16 results for "TGF-beta Receptor Inhibitors" in Products

TGF-beta Receptor Inhibitors

Potent, selective inhibitor of TGF-βRI, ALK4 and ALK7

GMP Version Available: TB1614-GMP
GMP
Chemical Name:
4-[4-(1,3-benzodioxol-5-yl)-5-(2-pyridinyl)-1H-imidazol-2-yl]benzamide
Purity:
≥99%
dopaminergic neurons derived from hiPSCs using SB 431542
(2)

SB 431542 synthesized to cGMP guidelines

Chemical Name:
4-[4-(1,3-benzodioxol-5-yl)-5-(2-pyridinyl)-1H-imidazol-2-yl]benzamide
Purity:
≥99%
SB 431542 synthesized to cGMP guidelines

Selective inhibitor of TGF-βRI, ALK4 and ALK7

Chemical Name:
3-(6-Methyl-2-pyridinyl)-N-phenyl-4-(4-quinolinyl)-1H-pyrazole-1-carbothioamide
Purity:
≥98%
Adult Stem Cell-derived Liver Organoids
(6)

Selective inhibitor of TGF-βRI

Chemical Name:
6-[2-(1,1-Dimethylethyl)-5-(6-methyl-2-pyridinyl)-1H-imidazol-4-yl]quinoxaline
Purity:
≥97%
Selective inhibitor of TGF-βRI

Selective inhibitor of TGF-βRI, ALK4 and ALK7

Chemical Name:
2-[4-(1,3-Benzodioxol-5-yl)-2-(1,1-dimethylethyl)-1H-imidazol-5-yl]-6-methyl-pyridine
Purity:
≥98%
Selective inhibitor of TGF-βRI, ALK4 and ALK7

Potent ATP-competitive TGF-βRI inhibitor

Chemical Name:
2-(5-Chloro-2-fluorophenyl)-4-[(4-pyridyl)amino]pteridine
Purity:
≥98%
Potent ATP-competitive TGF-βRI inhibitor

Potent and selective inhibitor of TGF-βRI

Chemical Name:
4-[4-[3-(2-Pyridinyl)-1H-pyrazol-4-yl]-2-pyridinyl]-N-(tetrahydro-2H-pyran-4-yl)-benzamide
Purity:
≥98%
Potent and selective inhibitor of TGF-βRI

RepSox synthesized to Ancillary Material Grade

Alternate Names:
ALK5 Inhibitor II,SJN 2511,E-616452
Chemical Name:
2-[3-(6-Methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,5-naphthyridine
Purity:
≥99%
RepSox synthesized to Ancillary Material Grade

Selective CK1 inhibitor. Also inhibits TGF-βRI

Chemical Name:
4-[4-(2,3-Dihydro-1,4-benzodioxin-6-yl)-5-(2-pyridinyl)-1H-imidazol-2-yl]benzamide
Purity:
≥98%
Selective CK1 inhibitor. Also inhibits TGF-βRI

ALK4 and ALK5 (TGFβRI) inhibitor

Alternate Names:
LY 2157299
Chemical Name:
4-[5,6-Dihydro-2-(6-methyl-2-pyridinyl)-4H-pyrrolo[1,2-b]pyrazol-3-yl]-6-quinolinecarboxamide
Purity:
≥98%
ALK4 and ALK5 (TGFβRI) inhibitor

Potent and selective inhibitor of TGF-βRI

Chemical Name:
4-[2-Fluoro-5-[3-(6-methyl-2-pyridinyl)-1H-pyrazol-4-yl]phenyl]-1H-pyrazole-1-ethanol
Purity:
≥98%
Potent and selective inhibitor of TGF-βRI

Potent and selective inhibitor of TGF-βRI

Chemical Name:
3-[[5-(6-Methyl-2-pyridinyl)-4-(6-quinoxalinyl)-1H-imidazol-2-yl]methyl]benzamide
Purity:
≥98%
Potent and selective inhibitor of TGF-βRI

Potent TGF-βRI inhibitor; orally bioavailable

Chemical Name:
4-[4-(1,3-Benzodioxol-5-yl)-5-(6-methyl-2-pyridinyl)-1H-imidazol-2-yl]bicyclo[2.2.2]octane-1-carboxamide
Purity:
≥98%
Potent TGF-βRI inhibitor; orally bioavailable

Potent TGF-βRI inhibitor

Chemical Name:
4-[[4-[(2.6-Dimethyl-3-pyridinyl)oxy]-2-pyridinyl]amino]benzenesulfonamide
Purity:
≥98%
Potent TGF-βRI inhibitor

Selective TGF-β kinase inhibitor

Chemical Name:
4-[5,6-Dihydro-2-(2-pyridinyl)-4H-pyrrolo[1,2-b]pyrazol-3-yl]-7-[2-(4-morpholinyl)ethoxy]quinoline
Purity:
≥98%
Selective TGF-β kinase inhibitor

Potent and selective inhibitor of TGF-βRI

Alternate Names:
E-616452,SJN 2511,ALK5 Inhibitor II
Chemical Name:
2-[3-(6-Methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,5-naphthyridine
Purity:
≥99%
Potent and selective inhibitor of TGF-βRI
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