7 results for "Histamine H4R Small Molecules and Peptides" in Products
Histamine H4R Small Molecules and Peptides
Histamine is a ubiquitous messenger molecule released from mast cells, enterochromaffin-like cells, and neurons. Its various actions are mediated by a family of histamine receptors, which are a subset of the G protein-coupled receptor superfamily. Histamine H4R is a histamine receptor that is predominantly expressed in hematopoietic cells. Histamine H4R is thought to play a role in inflammation and allergy reponses.
Selective, high affinity H4 agonist
H3 antagonist; also H4 inverse agonist
Standard H3 agonist. Also H4 agonist
Selective H4 antagonist
Selective H4 antagonist; orally active
Non-selective 5-HT, dopamine, adrenalin and histamine receptor antagonist; antipsychotic agent
High affinity and selective histamine H4 antagonist; orally bioavailable
