Skip to main content

94 results for "c-Abl" in Products

c-Abl Products

c-Abl (Abelson murine leukemia viral homolog 1) is a cytosolic member of the ABL subfamily, protein tyrosine kinase family of enzymes. It is ubiquitously expressed, and participates in multiple processes such as cell migration, actin reorganization, DNA damage response and apoptosis. Human c-Abl (I-B) is 1149 amino acids (aa) in length. It is myristoylated on Gly2 and contains one SH3 domain (aa 80-140), an SH2 domain (aa 146-236), a protein kinase region (aa 261-512), three NLS's (aa 620-634; ...

Show More

Potent, selective Src family kinase inhibitor

Chemical Name: 1-(1,1-Dimethylethyl)-1-(4-methylphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
Purity: ≥98% (HPLC)
Potent, selective Src family kinase inhibitor

Potent and selective Src tyrosine kinase family inhibitor; anticancer; antiviral; orally bioavailable

Alternate Names: AZD 0530
Chemical Name: N-(5-Chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methyl-1-piperazinyl)ethoxy]-5-[(tetrahydro-2H-pyran-4-yl)oxy]-4-quinazolinamine
Purity: ≥98% (HPLC)
Potent and selective Src tyrosine kinase family inhibitor; anticancer; antiviral; orally bioavailable

Highly potent pan-Src/Bcr-Abl inhibitor

Alternate Names: BMS-354825
Chemical Name: N-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-methyl-4-pyrimidinyl]amino]-5-thiazolecarboxamide
Purity: ≥98% (HPLC)
Highly potent pan-Src/Bcr-Abl inhibitor

Potent and selective v-Abl tyrosine kinase inhibitor; also inhibits PDGFR and c-kit

Alternate Names: Gleevec,CGP 57148B
Chemical Name: 4-[(4-Methyl-1-piperazinyl)methyl]-N-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]benzamide methanesulfonate
Purity: ≥98% (HPLC)
Potent and selective v-Abl tyrosine kinase inhibitor; also inhibits PDGFR and c-kit

Dual Src-Abl inhibitor; antiproliferative

Alternate Names: SKI-606
Chemical Name: 4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methyl-1-piperazinyl)propoxy]-3-quinolinecarbonitrile
Purity: ≥98%
Dual Src-Abl inhibitor; antiproliferative

Potent inhibitor of Abl T315l mutant and wild-type Abl kinases

Chemical Name: 5-[3-(2-Methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]-N,N-dimethyl-3-pyridinecarboxamide
Purity: ≥98% (HPLC)
Potent inhibitor of Abl T315l mutant and wild-type Abl kinases
Source: E. coli
Accession #: P00519.4
Applications: EnzAct

Potent multi-kinase and pan-Bcr-Abl inhibitor

Alternate Names: Ponatinib
Chemical Name: 3-(2-Imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N-[4-[(4-methyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-benzamide
Purity: ≥98% (HPLC)
Potent multi-kinase and pan-Bcr-Abl inhibitor

Src family kinase inhibitor; also inhibits c-Abl

Alternate Names: 1-NA-PP 1
Chemical Name: 1-(1,1-Dimethylethyl)-3-(1-naphthalenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
Purity: ≥98% (HPLC)
Src family kinase inhibitor; also inhibits c-Abl

Selective allosteric inhibitor of Bcr-Abl; analog of GNF 2 (Cat. No. 4399)

Chemical Name: N-(2-Hydroxyethyl)-3-[6-[[4-(trifluoromethoxy)phenyl]amino]-4-pyrimidinyl]benzamide
Purity: ≥98% (HPLC)
Selective allosteric inhibitor of Bcr-Abl; analog of GNF 2 (Cat. No. 4399)

BCR-ABL1 kinase PROTAC® Degrader

Chemical Name: (2S,4R)-1-((S)-3,3-Dimethyl-2-(2-(2-(4-(6-((4-(trifluoromethoxy)phenyl)amino)pyrimidin-4-yl)phenoxy)ethoxy)acetamido)butanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity: ≥98% (HPLC)
BCR-ABL1 kinase PROTAC®

Ras signaling inhibitor; inhibits Ack1 and GCK

Chemical Name: N-[3-[1,4-Dihydro-1-methyl-7-[(6-methyl-3-pyridinyl)amino]-2-oxopyrimido[4,5-d]pyrimidin-3(2H)-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide
Purity: ≥98% (HPLC)
Ras signaling inhibitor; inhibits Ack1 and GCK

Potent EGFR and VEGFR inhibitor

Chemical Name: 6-[4-[(4-Ethyl-1-piperazinyl)methyl]phenyl]-N-[(1R)-1-phenylethyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
Purity: ≥98% (HPLC)
Potent EGFR and VEGFR inhibitor
Reactivity: Human, Mouse
Details: Mouse IgG1 Monoclonal Clone #8E9
Applications: IHC, WB, ICC/IF, IP
Western Blot: c-Abl Antibody (8E9) [NBP2-49695]
(3)
Reactivity: Human
Details: Rabbit IgG Polyclonal
Applications: IHC, WB, ICC/IF
Western Blot: c-Abl Antibody [NBP2-15631]
(4)
Reactivity: Human
Details: Rabbit IgG Polyclonal
Applications: IHC, ICC/IF
Immunocytochemistry/ Immunofluorescence: c-Abl Antibody [NBP1-90289]
(2)
Results Per Page
5 10 25 50
/ 4