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CE3F4

Tocris Bioscience, part of Bio-Techne | Catalog # 4793

Noncompetitive Epac1 inhibitor
Discontinued Product
4793 has been discontinued. View all EPAC Inhibitors products.

Key Product Details

Description

Noncompetitive Epac1 inhibitor

Product Description

CE3F4 is a noncompetitive Epac1 inhibitor. Blocks Epac-induced Rap activation and prevents isoprenaline-induced autophagy flux in cardiomyocytes. Has no effect on PKA activity in the presence of cAMP.

Product Specifications

Molecular Weight

351.01

Formula

C11H10Br2FNO

Storage

Store at -20°C

Purity

≥98% (HPLC)

Chemical Name

5,7-Dibromo-6-fluoro-3,4-dihydro-2-methyl-1(2H)-quinolinecarboxaldehyde

CAS Number

143703-25-7

PubChem ID

21781066

InChI Key

ZZLQPWXVZCPUGC-UHFFFAOYSA-N

SMILES

BrC1=C(F)C(Br)=C(CCC(C)N2C=O)C2=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 35.1 100
Ethanol 17.55 50

Preparing Stock Solutions for CE3F4

The following data is based on the product molecular weight 351.01

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.85 mL 14.24 mL 28.49 mL
5 mM 0.57 mL 2.85 mL 5.70 mL
10 mM 0.28 mL 1.42 mL 2.85 mL
50 mM 0.06 mL 0.28 mL 0.57 mL

Calculators

Molarity Calculator

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Dilution Calculator

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Reconstitution Calculator

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Background References

References are publications that support the biological activity of the product.

Product Documents for CE3F4

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for CE3F4

For research use only

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