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56 results for "e3 ligase inhibitors" in Products

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56 results for "e3 ligase inhibitors" in Products

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Catalog #: 6466

Carboxylic acid-functionalized Thalidomide; cereblon ligand for PROTACs

Chemical Name : 2-[[2-(2,6-Dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]acetic acid
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule
Catalog #: 6945

Potent and selective (+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo

Chemical Name : (6S)-4-(4-Chlorophenyl)-N-[8-[[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]acetyl]amino]octyl]-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide
Purity : ≥98% (HPLC)
Active Degraders Small Molecule

HECT E3 ubiquitin ligase inhibitor

Chemical Name : N-(4-Acetylphenyl)-3-(5-ethyl-2-furanyl)-2-propenamide
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule
Catalog #: 5636

β-TrCP1 ligase inhibitor

Chemical Name : 4-[4-[[5-(2-Fluorophenyl)-2-furanyl]methylene]-4,5-dihydro-5-oxo-3-(phenylmethyl)-1H-pyrazol-1-yl]benzoic acid
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule
Catalog #: 6305

Cereblon binder; induces ubiquitination and degradation of CK1α by E3 ubiquitin ligase

Chemical Name : 3-(4-Amino-1,3-dihydro-1-oxo-2H-isoindol-2-yl)-2,6-piperidinedione
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule

(+)-JQ1 based Degrader (PROTAC®) that selectively degrades BRD4

Chemical Name : (2S,4R)-1-((S)-2-(tert-butyl)-17-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,16-dioxo-6,9,12-trioxa-3,15-diazaheptadecanoyl)- 4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity : ≥98% (HPLC)
Active Degraders Small Molecule
Catalog #: 6782

Molecular glue; pre-mRNA splicing modulator

Chemical Name : N1-(3-Chloro-1H-indol-7-yl)-1,4-benzenedisulfonamide
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule

Selective Skp2 inhibitor; suppresses E3 ligase activity

Chemical Name : 3-(2-Benzothiazolyl)-6-ethyl-7-hydroxy-8-(1-piperidinylmethyl)-4H-1-benzopyran-4-one
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule

Functionalized VHL ligand for PROTACs

Chemical Name : (4R)-3-Methyl-L-valyl-4-hydroxy-N-[[4-(4-methyl-5-thiazolyl)phenyl]methyl]-L-prolinamide dihydrochloride
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule
Catalog #: 6327

(+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo

Chemical Name : (6S)-4-(4-Chlorophenyl)-N-[4-[[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]acetyl]amino]butyl]-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide
Purity : ≥98% (HPLC)
Active Degraders Small Molecule
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