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53 results for "e3 ligase inhibitors" in Products

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53 results for "e3 ligase inhibitors" in Products

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HECT E3 ubiquitin ligase inhibitor

Chemical Name : N-(4-Acetylphenyl)-3-(5-ethyl-2-furanyl)-2-propenamide
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule
Catalog #: 4375

Selective inhibitor of E3 ubiquitin ligase

Chemical Name : 9H-Indeno[1,2-e][1,2,5]oxadiazolo[3,4-b]pyrazin-9-one
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule
Catalog #: 6466

Carboxylic acid-functionalized Thalidomide; cereblon ligand for PROTACs

Chemical Name : 2-[[2-(2,6-Dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]acetic acid
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule
Catalog #: 6327

(+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo

Chemical Name : (6S)-4-(4-Chlorophenyl)-N-[4-[[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]acetyl]amino]butyl]-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide
Purity : ≥98% (HPLC)
Active Degraders Small Molecule
Catalog #: 5636

β-TrCP1 ligase inhibitor

Chemical Name : 4-[4-[[5-(2-Fluorophenyl)-2-furanyl]methylene]-4,5-dihydro-5-oxo-3-(phenylmethyl)-1H-pyrazol-1-yl]benzoic acid
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule
Catalog #: 6305

Cereblon binder; induces ubiquitination and degradation of CK1α by E3 ubiquitin ligase

Chemical Name : 3-(4-Amino-1,3-dihydro-1-oxo-2H-isoindol-2-yl)-2,6-piperidinedione
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule

(+)-JQ1 based Degrader (PROTAC®) that selectively degrades BRD4

Chemical Name : (2S,4R)-1-((S)-2-(tert-butyl)-17-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,16-dioxo-6,9,12-trioxa-3,15-diazaheptadecanoyl)- 4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity : ≥98% (HPLC)
Active Degraders Small Molecule

Inhibitor of Bmi1/Ring1A; blocks histone H2A ubiquitination

Chemical Name : 2-(3-Pyridinylmethylene)-1H-Indene-1,3(2H)-dione
Purity : ≥99% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule

Cdc20 inhibitor; inhibits Cdc20-substrate interaction

Chemical Name : 3-(2-Methyl-5-nitroimidazol-1-yl)-N-(2,2,2-trichloro-1-phenylaminoethyl)propionamide
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule

Functionalized VHL ligand for PROTACs

Chemical Name : (4R)-3-Methyl-L-valyl-4-hydroxy-N-[[4-(4-methyl-5-thiazolyl)phenyl]methyl]-L-prolinamide dihydrochloride
Purity : ≥98% (HPLC)
Ubiquitin Ligase (E3) Inhibitors Small Molecule
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