ICI 154,129

Name: ICI 154,129
Brand: tocris
SKU: 0827

Catalog # 0827

Citations (1)

Datasheet / COA / SDS

Order Information

Bio-Techne Corporation

tel: (800) 343-7475 (free phone)

tel: (612) 379-2956

customercare.na@bio-techne.com

Shipping Information

$35 to United States

Products in stock will be shipped in 1-3 business days unless specified.

View Distributors

Key Product Details

Description:	δ selective peptide antagonist
Molecular Weight:	638.83

View Full Technical Details for ICI 154,129

Biological Activity

ICI 154,129 is a selective δ opioid antagonist.

Licensing Information

Sold with the permission of AstraZeneca UK Ltd.

Technical Data

M. Wt	638.83
Formula	C₃₄H₄₆N₄O₆S
Single Letter Sequence	YGFL (Modifications: Tyr-1 = N,N-diallyl-Tyr, Gly-2 - Phe-3 peptide bond replaced with Psi-(CH₂S))
Storage	Desiccate at -20°C
CAS Number	83420-94-4
PubChem ID	3035055
InChi Key	CZRZYRKTYLLLRL-DTXPUJKBSA-N
Smiles	CC(C)C[C@H](NC(=O)[C@H](CC1=CC=CC=C1)SCCNC(=O)CNC(=O)[C@H](CC1=CC=C(O)C=C1)N(CC=C)CC=C)C(O)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Solubility

Soluble to 1mg in methanol

Molarity Calculator

Calculate the mass, volume, or concentration required for a solution.

Mass

Concentration

Volume

M. Wt*

g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and CoA (available online).

Dilution Calculator

Calculate the dilution required to prepare a stock solution.

Concentration 1 (C1)

Volume 1 (V1)

Concentration 2 (C2)

Volume 2 (V2)

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

Volume (to add to vial)

Mass (in vial)

Desired Reconstitution Concentration

References

References are publications that support the biological activity of the product.

Shaw Selective antagonists at the opiate delta-receptor. Life Sci. 1982 PMID: 6128652
Rees and Hunter Opioid Receptors. Comprehensive Medicinal Chemistry. Ed. Hansch.

Citations (1)

Showing 1 - 1 of 1 citation Showing All

Search Title:

Citations are publications that use Bio-Techne products. Selected citations for ICI 154,129 include:

Jiang et al. (2015) Analgesic roles of peripheral intrinsic met-enkephalin and dynorphin A in long-lasting inflammatory pain induced by complete Freund's adjuvant in rats. J Pharmacol Exp Ther. 9:2344
PMID: 26136984

There are no citations that match your criteria.

Showing 1 - 1 of 1 citation Showing All

Product Datasheets

COA

Certificate of Analysis is currently unavailable on-line. Please contact Customer Service.

ICI 154,129

Order Information

Shipping Information

Key Product Details

Complete Your Experiment

Biological Activity

Licensing Information

Technical Data

Solubility

Molarity Calculator

Dilution Calculator

Reconstitution Calculator

References

Citations (1)

Product Datasheets

COA

SDS

Bio-Techne Brands

Stay Connected