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5 results for "Tankyrase Inhibitors Small Molecules and Peptides" in Products

Tankyrase Inhibitors Small Molecules and Peptides

Potent tankyrase inhibitor

GMP Version Available: TB3748-GMP
GMP
Alternate Names:
XAV939 Wnt Signaling Inhibitor
Chemical Name:
3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one
Purity:
≥98%
Potent tankyrase inhibitor

XAV 939 synthesized to cGMP guidelines

Chemical Name:
3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one
Purity:
≥99%
XAV 939 synthesized to cGMP guidelines

Potent TNKS1/2 inhibitor

Chemical Name:
rel-2-[4-[6-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]-4-methyl-3-pyridinyl]phenyl]-3,7-dihydro-7-methyl-4H-pyrrolo[2,3-d]pyrimidin-4-one
Purity:
≥98%
Potent TNKS1/2 inhibitor

Potent tankyrase inhibitor

Chemical Name:
2-[3-[[4-(4-Methoxyphenyl)-5-(4-pyridinyl)-4H-1,2,4-triazol-3-yl]thio]propyl]-1H-benz[de]isoquinoline-1,3(2H)-dione
Purity:
≥98%
Potent tankyrase inhibitor

Potent tankyrase inhibitor

Chemical Name:
2-[3-[[4-(4-Methoxyphenyl)-5-(4-pyridinyl)-4H-1,2,4-triazol-3-yl]thio]propyl]-1H-benz[de]isoquinoline-1,3(2H)-dione
Purity:
≥98%
Potent tankyrase inhibitor
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