Brg1: Small Molecules and Peptides
4 results for "Brg1 Small Molecules and Peptides" in Products
4 results for "Brg1 Small Molecules and Peptides" in Products
Brg1: Small Molecules and Peptides
BRG1/SMARCA4 Degrader (PROTAC®)
| Chemical Name: | 3-((4-(3-(2-Chloropyridin-4-yl)ureido)pyridin-2-yl)ethynyl)-N-(4-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)butyl)benzamide |
| Purity: | ≥95% (HPLC) |
Potent and selective SMARCA4/2 inhibitor
| Chemical Name: | (S)-1-(Methylsulfonyl)-N-[4-(methylthio)-1-oxo-1-[[4-[3-(pyridin-4-yl)phenyl]thiazol-2-yl]amino]butan-2-yl]-1H-pyrrole-3-carboxamide |
| Purity: | ≥95% (HPLC) |
Potent SMARCA2/4 inhibitor
| Chemical Name: | N-[(1S)-1-(Methoxymethyl)-2-[[4-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]-2-thiazolyl]amino]-2-oxoethyl]-1-(methylsulfonyl)-1H-pyrrole-3-carboxamide |
| Purity: | ≥95% (HPLC) |
Potent and selective SMARCA2/4 and polybromo 1 inhibitor
| Chemical Name: | (2E)-1-(2-Hydroxyphenyl)-3-[(1R,4R)-5-(pyridin-2-yl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]prop-2-en-1-one |
| Purity: | ≥98% (HPLC) |