PSB 1114

Name: PSB 1114
Brand: Tocris Bioscience
SKU: 4333

Tocris Bioscience, part of Bio-Techne | Catalog # 4333

Citations (7)

COA / SDS

Potent, selective P2Y2 agonist

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Product Description
Product Specifications
Solubility
Calculators
Background References
Product Documents
Specific Notices

Key Product Details

Description

Potent, selective P2Y2 agonist

View all P2Y Receptor Agonists »

Product Description

PSB 1114 is a potent, selective P2Y₂ agonist (EC₅₀ = 0.134 μM). Displays >60-fold selectivity versus P2Y₄ and P2Y₆ receptors.

Product Specifications

Molecular Weight

622.14

Formula

C₁₀H₁₁F₂N₂Na₄O₁₃P₃S

Storage

Store at -80°C

Purity

≥98% (HPLC)

Chemical Name

4-Thiouridine-5'-O-(β,γ-difluoromethylene)triphosphate tetrasodium salt

CAS Number

1657025-60-9

PubChem ID

90488930

InChI Key

KATPYMNMKKBLAH-GENVZAMMSA-J

SMILES

[Na+].[Na+].[Na+].[Na+].O[C@H]1[C@@H](O)C(O[C@@H]1COP([O-])(=O)OP([O-])(=O)C(F)(F)P([O-])([O-])=O)N1C=CC(=S)NC1=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Soluble in water (supplied pre-dissolved at a concentration of 10mM)

Calculators

Molarity Calculator

Calculate the mass, volume, or concentration required for a solution.

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*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and CoA (available online).

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Reconstitution Calculator

Background References

References are publications that support the biological activity of the product.

El-Tayeb Structural modifications of UMP, UDP, and UTP leading to subtype-selective agonists for P2Y₂, P2Y₄, and P2Y₆ receptors. J.Med.Chem. 2011 PMID: 21417463